SCHEMBL8429158

SCHEMBL8429158

NN([C@](C(=O)O)(C(=C=O)c1ccccc1)c1cccc(NC2=NCCN2)c1)S(=O)(=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.44
ITGAV P06756 13/20 0.44
ITGA2B P08514 12/20 0.44
ITGB1 P05556 5/20 0.41
ITGB5 P18084 5/20 0.41
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
PTGIR P43119 2/20 0.34
F2 P00734 1/20 0.34
C1R P00736 1/20 0.34
F10 P00742 1/20 0.34
KLKB1 P03952 1/20 0.34
KLK1 P06870 1/20 0.34
PRSS1 P07477 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8430880 0.78 CA1 (0.37) F2
SCHEMBL8430809 0.71 CA1 (0.32)
SCHEMBL8696196 0.70 ITGB3 (0.48) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL7753126 0.69 ADRA2A (0.58) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8432276 0.68 ITGB3 (0.33) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8429290 0.68 CA1 (0.33)
Hydrochloric Acid SCHEMBL7562956 0.68 ADRA2A (0.57) ITGB3ITGAVITGA2BITGB1ITGB5
Benzophenone SCHEMBL5084127 0.66 ADRA2A (0.80) ITGB3ITGAVITGA2BITGB1ITGB5
SCHEMBL8431435 0.64 CA1 (0.32)
SCHEMBL1036359 0.63 ADRA2A (0.78) ADRA2AADRA2BADRA2CPTGIR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed