SCHEMBL8429321

SCHEMBL8429321

NN=CNc1cccc(C(=O)c2ccc(CCC(=O)O)c(CCC(=O)O)c2N)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.38
ITGA2B P08514 6/20 0.38
ITGAV P06756 4/20 0.38
FOS P01100 1/20 0.35
JUN P05412 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
LTB4R Q15722 1/20 0.33
ITGB1 P05556 1/20 0.32
ITGB5 P18084 1/20 0.32
SIRT1 Q96EB6 1/20 0.32
ABCB11 O95342 1/20 0.32
LMNA P02545 1/20 0.32
PTGS1 P23219 1/20 0.32
ADORA1 P30542 1/20 0.32
PTGS2 P35354 1/20 0.32
PTGER1 P34995 1/20 0.32
PTGER4 P35408 1/20 0.32
PTGER3 P43115 1/20 0.32
PTGER2 P43116 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8431244 0.94 ITGB3 (0.37) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8432903 0.89 ITGB3 (0.39) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8429187 0.89 ITGB3 (0.37) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8432521 0.88 ABCB11 (0.41) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8428908 0.88 ITGB3 (0.38) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8432815 0.86 ITGB3 (0.40) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8532340 0.83 PTGS1 (0.39) CA1CA2ABCB11LMNAPTGS1
SCHEMBL8532447 0.80 PTGS1 (0.40) CA1CA2ABCB11LMNAPTGS1
SCHEMBL8429208 0.80 SIRT1 (0.37) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8530525 0.79 ABCB11 (0.54) CA1CA2ABCB11LMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed