SCHEMBL8428908

SCHEMBL8428908

NN=CNc1cccc(C(=O)c2ccc(CCC(=O)O)c(N)c2O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.38
ITGA2B P08514 6/20 0.38
ITGAV P06756 4/20 0.38
FOS P01100 1/20 0.35
JUN P05412 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
HSD17B14 Q9BPX1 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
RECQL P46063 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ITGB1 P05556 1/20 0.32
ITGB5 P18084 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8432521 0.88 ABCB11 (0.41) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8429321 0.88 ITGB3 (0.38) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8429187 0.87 ITGB3 (0.37) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8432903 0.87 ITGB3 (0.39) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8431244 0.86 ITGB3 (0.37) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8432815 0.84 ITGB3 (0.40) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8429208 0.80 SIRT1 (0.37) ITGB3ITGA2BITGAVFOSJUN
SCHEMBL8698661 0.79 KDM4E (0.38) ITGB3ITGA2BITGAVCA1CA2
SCHEMBL8532447 0.78 PTGS1 (0.40) CA1CA2MEN1KMT2AFFAR1
SCHEMBL8532340 0.77 PTGS1 (0.39) CA1CA2KDM4EMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed