SCHEMBL8429381

SCHEMBL8429381

COCc1ccc(COC(Cl)c2ccc(COC)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.38
AOC3 Q16853 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
ATM Q13315 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
ACACB O00763 1/20 0.33
PTGS2 P35354 1/20 0.32
ESR1 P03372 2/20 0.32
ESR2 Q92731 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
ADRB3 P13945 1/20 0.32
AGXT P21549 2/20 0.31
PPARG P37231 2/20 0.30
PPARA Q07869 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9319276 0.81 IDO1 (0.42) IDO1L3MBTL1TSHRMAPK1ATM
SCHEMBL11307378 0.76 IDO1 (0.45) IDO1L3MBTL1ACACBPTGS2ESR1
SCHEMBL28528002 0.76 CHRNB2 (0.45) CHRNB2CHRNA4CYP2C19AGXTSLC6A2
SCHEMBL547986 0.75 SLC6A2 (0.47) IDO1AOC3TSHRTDP1CHRNB2
SCHEMBL134443 0.75 IDO1 (0.46) IDO1TSHRACACBPTGS2AGXT
SCHEMBL11875424 0.74 ALDH1A1 (0.46) TSHRATMCYP1A2CYP2D6
SCHEMBL764954 0.74 IDO1 (0.65) IDO1L3MBTL1ACACBESR1ESR2
SCHEMBL12134040 0.74 ACACB (0.39) IDO1L3MBTL1ACACBPTGS2ADRB3
SCHEMBL6181884 0.73 CHRNB2 (0.63) IDO1MAPK1TDP1CHRNB2CHRNA4
SCHEMBL8954887 0.72 IDO1 (0.42) IDO1L3MBTL1ACACBPTGS2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877321-A NEUROKININ RECEPTOR SANOFI (FR) 1999-03-02 US disclosed
US-5446052-A Used for treatment of substance p-and neurokinin-dependent pathology such as analgesia and inflmmation SANOFI (FR) 1995-08-29 US disclosed
US-5300648-A Analgesics, antiinflammatory agents SOCIETE ANONYME: ELF SANOFI (FR) 1994-04-05 US disclosed