SCHEMBL8429467

SCHEMBL8429467

NN=CNc1cccc(C(=O)C(C(=O)O)C(N)(C(=O)O)c2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 1/20 0.41
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA4 P22748 1/20 0.34
LMNA P02545 1/20 0.33
KMT2A Q03164 5/20 0.33
MEN1 O00255 4/20 0.33
NPC1 O15118 3/20 0.33
MAPT P10636 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
ALDH1A1 P00352 2/20 0.33
NFKB1 P19838 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
GAA P10253 2/20 0.33
RAB9A P51151 2/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8431264 0.74 CA1 (0.36) CA1CA2CA4LMNAKMT2A
SCHEMBL6777725 0.73 RAB9A (0.50) CA1CA2KMT2AMEN1NPC1
SCHEMBL8429166 0.70 CA1 (0.43) CA1CA2CA4KMT2AMEN1
SCHEMBL8429109 0.70 MEN1 (0.37) CYP1A2CA1CA2CA4KMT2A
SCHEMBL8542413 0.69 KCNK3 (0.41) CA1CA2CA4LMNAKMT2A
SCHEMBL8431435 0.68 CA1 (0.32) CA1CA2CA4LMNAKMT2A
SCHEMBL8532972 0.68 KMT2A (0.33) CYP1A2KMT2AMEN1NPC1MAPT
SCHEMBL8432262 0.68 ERCC5 (0.38) CYP1A2CA1CA2CA4KMT2A
SCHEMBL8430799 0.68 SIRT2 (0.41) KMT2AMEN1SMN1; SMN2ALDH1A1TP53
SCHEMBL8697026 0.67 CA1 (0.40) CA1CA2CA4KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed