SCHEMBL8430799

SCHEMBL8430799

NN=CNc1cccc(C(=O)N(N)[C@@H](Cc2ccccc2)C(=O)O)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ADORA2A P29274 1/20 0.38
GPR132 Q9UNW8 1/20 0.36
SLC7A5 Q01650 3/20 0.36
ALPI P09923 1/20 0.36
PKM P14618 1/20 0.36
PTGS1 P23219 1/20 0.36
XIAP P98170 1/20 0.36
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
TP53 P04637 1/20 0.35
ROCK2 O75116 1/20 0.35
GRK2 P25098 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7380583 0.85 GPR132 (0.39) ALDH1A1SMN1; SMN2GPR132SLC7A5
SCHEMBL7380590 0.85 GPR132 (0.39) ALDH1A1SMN1; SMN2GPR132SLC7A5
SCHEMBL7376071 0.82 ITGB3 (0.39) MEN1KMT2AALDH1A1GPR132SLC7A5
SCHEMBL7376076 0.82 ITGB3 (0.39) MEN1KMT2AALDH1A1GPR132SLC7A5
SCHEMBL7375578 0.81 ALDH1A1 (0.41) MEN1KMT2AALDH1A1SMN1; SMN2GPR132
SCHEMBL7375584 0.81 ALDH1A1 (0.41) MEN1KMT2AALDH1A1SMN1; SMN2GPR132
SCHEMBL7375604 0.81 ALDH1A1 (0.39) MEN1KMT2AALDH1A1SMN1; SMN2GPR132
SCHEMBL7375609 0.81 ALDH1A1 (0.39) MEN1KMT2AALDH1A1SMN1; SMN2GPR132
SCHEMBL7466500 0.79 ITGB3 (0.40) MEN1KMT2AALDH1A1SMN1; SMN2GPR132
SCHEMBL7409609 0.79 ALDH1A1 (0.38) MEN1KMT2AALDH1A1SMN1; SMN2GPR132

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed