SCHEMBL8430946

SCHEMBL8430946

NN=CNc1cccc(C(=O)c2ccc(CC(=O)O)c(Oc3ccccc3)c2N)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.39
ABCB11 O95342 1/20 0.36
LMNA P02545 1/20 0.36
PTGS1 P23219 1/20 0.36
ADORA1 P30542 1/20 0.36
PTGS2 P35354 1/20 0.36
CAMK2A Q9UQM7 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
FFAR1 O14842 1/20 0.35
STS P08842 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
NR1H4 Q96RI1 1/20 0.34
ERCC5 P28715 1/20 0.34
FEN1 P39748 1/20 0.34
FABP1 P07148 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8532447 0.83 PTGS1 (0.40) SRD5A2ABCB11LMNAPTGS1ADORA1
SCHEMBL8530525 0.82 ABCB11 (0.54) ABCB11LMNAPTGS1ADORA1PTGS2
SCHEMBL8532340 0.82 PTGS1 (0.39) ABCB11LMNAPTGS1ADORA1PTGS2
SCHEMBL8432815 0.79 ITGB3 (0.40) LMNAMEN1KMT2AFFAR1ALDH1A1
SCHEMBL8429321 0.76 ITGB3 (0.38) ABCB11LMNAPTGS1ADORA1PTGS2
SCHEMBL8432903 0.75 ITGB3 (0.39) SRD5A2ABCB11LMNAPTGS1ADORA1
SCHEMBL8429187 0.75 ITGB3 (0.37) FFAR1CA1CA2
SCHEMBL8431244 0.74 ITGB3 (0.37) PTGS1PTGS2FFAR1CA1CA2
SCHEMBL8432521 0.74 ABCB11 (0.41) ABCB11LMNAPTGS1ADORA1PTGS2
SCHEMBL8428908 0.74 ITGB3 (0.38) SRD5A2MEN1KMT2AFFAR1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed