SCHEMBL8430969

SCHEMBL8430969

CC(C)(C)CC(=O)N(N)[C@](C(=O)O)(C(=C=O)c1ccccc1)c1cccc(NC=NN)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 3/20 0.33
KCNK9 Q9NPC2 1/20 0.32
CYP2C19 P33261 5/20 0.31
CYP3A4 P08684 3/20 0.31
CYP2C9 P11712 3/20 0.31
HPGD P15428 2/20 0.31
RAB9A P51151 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP1A2 P05177 2/20 0.31
HDAC3 O15379 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8429207 0.89 P2RX1 (0.36) CYP2C19CYP3A4CYP2C9HPGDCYP1A2
SCHEMBL8431435 0.87 CA1 (0.32) RAB9AKMT2ASMN1; SMN2LMNAHTT
SCHEMBL8429055 0.86 TRPV4 (0.35) KCNK9CYP2C19CYP3A4KMT2ACYP1A2
SCHEMBL8431235 0.86 RXFP1 (0.32) KCNK9CYP2C19CYP3A4RAB9AKMT2A
SCHEMBL8429290 0.83 CA1 (0.33) KCNK9CYP2C19CYP3A4RAB9AKMT2A
SCHEMBL8430960 0.83 MAPT (0.35) CYP2C19CYP3A4HPGDRAB9AKMT2A
SCHEMBL8432441 0.83 KMT2A (0.32) RAB9AKMT2ACYP1A2SMN1; SMN2LMNA
SCHEMBL8429159 0.82 NR1H4 (0.32) NR1H4HPGDRAB9AKMT2AALDH1A1
SCHEMBL8432619 0.81 TRPV4 (0.35) HPGDRAB9AALDH1A1MAPT
SCHEMBL8521199 0.81 ALDH1A1 (0.36) HPGDRAB9AKMT2ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US claimed
US-5952381-A SELECTIVELY INHIBITING OR ANTAGONIZING THE INTEGRINS; ANTITUMOR AGENTS, ANTIARTHRITIC AGENTS, VIRICIDES, MICROBIOCIDES; TREATING OSTEOPOROSIS, SKIN DISORDERS G. D. SEARLE & CO. (US) 1999-09-14 US disclosed