SCHEMBL8433873

SCHEMBL8433873

CCOC(=O)/C(Cc1c[nH]c2ccc(Br)cc12)=N/O

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.53
GABRB1 P18505 1/20 0.53
GABRA3 P34903 1/20 0.53
GABRB2 P47870 1/20 0.53
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
GPR84 Q9NQS5 1/20 0.48
PKM P14618 1/20 0.46
NR4A2 P43354 1/20 0.44
HTR2A P28223 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.44
CSNK2A1 P68400 1/20 0.43
KDM4E B2RXH2 1/20 0.43
SLC6A4 P31645 1/20 0.43
SIGMAR1 Q99720 1/20 0.42
IDO1 P14902 1/20 0.42
ICMT O60725 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3849942 1.00 GABRA1 (0.53) GABRA1GABRB1GABRA3GABRB2MTNR1A
SCHEMBL3849939 1.00 GABRA1 (0.53) GABRA1GABRB1GABRA3GABRB2MTNR1A
SCHEMBL13333453 0.91 GABRA1 (0.53) GABRA1GABRB1GABRA3GABRB2MTNR1A
SCHEMBL17520646 0.87 NPSR1 (0.56) PKMHTR2AKDM4ESLC6A4IDO1
SCHEMBL24012125 0.85 KDM4E (0.62) MTNR1AMTNR1BGPR84HTR2ATRPM8
SCHEMBL17500189 0.85 KDM4E (0.62) MTNR1AMTNR1BGPR84HTR2ATRPM8
SCHEMBL7956840 0.83 PKM (0.67) PKMKDM4E
SCHEMBL7956839 0.83 PKM (0.67) PKMKDM4E
SCHEMBL8442871 0.83 PKM (0.67) PKMKDM4E
SCHEMBL3703101 0.83 PKM (0.67) GABRA1GABRB1GABRA3GABRB2MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1964835-A1 Derivatives of psammaplin A, a method for their synthesis and their use for the prevention or treatment of cancer Centre National de la Recherche Scientifique (FR) 2008-09-03 EP disclosed