SCHEMBL8433930

SCHEMBL8433930

CCC1CCN(C(=O)N(CCN2CCC(c3ccccc3OC)CC2)c2ccccn2)CC1.CCC1CCN(C(=O)OC(Cl)(Cl)Cl)CC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.46
ADRA1A P35348 4/20 0.46
DRD4 P21917 3/20 0.46
ADRA1D P25100 3/20 0.46
ADRA1B P35368 3/20 0.46
CYP2D6 P10635 3/20 0.46
TSHR P16473 2/20 0.46
CYP3A4 P08684 2/20 0.46
HTR1B P28222 1/20 0.46
HTR7 P34969 1/20 0.46
HTR2B P41595 1/20 0.46
OPRM1 P35372 1/20 0.45
CYP2C19 P33261 1/20 0.45
MTOR P42345 1/20 0.45
RAB9A P51151 1/20 0.45
HIF1A Q16665 1/20 0.45
DRD2 P14416 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27510623 0.92 OPRM1 (0.51) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL8298272 0.84 HTR1A (0.56) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL8303894 0.83 HTR1A (0.57) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL8299404 0.83 HTR1A (0.57) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL8303685 0.83 HTR1A (0.50) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL8298214 0.79 HTR1A (0.54) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL8304236 0.78 HTR1A (0.53) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL8297779 0.75 HTR1A (0.75) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL27532215 0.75 DRD2 (0.52) HTR1AADRA1ADRD4ADRA1DADRA1B
SCHEMBL8297150 0.71 HTR1A (0.71) HTR1AADRA1ADRD4ADRA1DADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0898569-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GmbH (DE) 1999-03-03 EP disclosed
WO-1997040038-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GMBH (DE) 1997-10-30 WO disclosed