SCHEMBL8435003

SCHEMBL8435003

CC(C)c1noc(C#N)c1OC(=O)NC1CC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
IDH1 O75874 4/20 0.32
SMYD3 Q9H7B4 2/20 0.32
HTT P42858 2/20 0.31
LMNA P02545 1/20 0.31
AR P10275 1/20 0.31
IRAK4 Q9NWZ3 2/20 0.31
ALDH1A1 P00352 1/20 0.30
CTSL P07711 1/20 0.30
CTSB P07858 1/20 0.30
CTSH P09668 1/20 0.30
CTSK P43235 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8436037 0.80 IDH1 (0.38) RAB9ANPC1TSHRSMN1; SMN2IDH1
SCHEMBL8440545 0.79 NPC1 (0.34) RAB9ANPC1TSHRSMN1; SMN2SMYD3
SCHEMBL9074668 0.78 NPC1 (0.43) RAB9ANPC1TSHRSMN1; SMN2SMYD3
SCHEMBL8441619 0.77
SCHEMBL9077785 0.70 NPC1 (0.43) RAB9ANPC1TSHRSMN1; SMN2IDH1
SCHEMBL8438552 0.69 SMN1; SMN2 (0.42) RAB9ANPC1TSHRSMN1; SMN2SMYD3
SCHEMBL3050719 0.64 MLYCD (0.30)
SCHEMBL9076104 0.62 NPC1 (0.42) RAB9ANPC1TSHRSMN1; SMN2SMYD3
SCHEMBL9077297 0.62 NPC1 (0.42) RAB9ANPC1TSHRSMN1; SMN2SMYD3
SCHEMBL8438550 0.61 NPC1 (0.45) RAB9ANPC1TSHRSMN1; SMN2SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0669326-B1 Cyanoisoxazoles BASF AG (DE) 1999-12-22 EP disclosed
EP-0669326-A1 Cyanoisoxazoles BASF Aktiengesellschaft (DE) 1995-08-30 EP disclosed