SCHEMBL8436353

SCHEMBL8436353

CC1CCc2ccc(NC(=O)NC3CCCC3)cc21.CCCNCCC

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.49
RAB9A P51151 9/20 0.49
SMN1; SMN2 Q16637 5/20 0.48
EPHX1 P07099 6/20 0.47
EPHX2 P34913 3/20 0.47
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
PKM P14618 1/20 0.45
ALOX15 P16050 1/20 0.45
TP53 P04637 2/20 0.44
NFKB1 P19838 2/20 0.44
NFKB2 Q00653 2/20 0.44
RELA Q04206 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8436872 0.86 MTNR1A (0.45) NPC1RAB9ASMN1; SMN2HTT
SCHEMBL8433416 0.84 MTNR1A (0.58) NPC1RAB9A
SCHEMBL8432113 0.83 NPC1 (0.49) NPC1RAB9ASMN1; SMN2EPHX1EPHX2
SCHEMBL8432869 0.82 EPHX1 (0.51) EPHX1EPHX2HTT
SCHEMBL8432637 0.81 MTNR1A (0.44) TSHR
SCHEMBL8432408 0.77 RAB9A (0.51) NPC1RAB9ASMN1; SMN2TP53NFKB1
SCHEMBL8436348 0.77 NPC1 (0.47) NPC1RAB9ASMN1; SMN2EPHX1EPHX2
SCHEMBL8436852 0.77 MTNR1A (0.38)
Oxalic Acid SCHEMBL8432169 0.76 MTNR1A (0.39)
SCHEMBL8697680 0.76 MTNR1A (0.36) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972964-A FOR TREATMENT OF CERTAIN PSYCHIC AND NEUROLOGIC DISORDERS SUCH AS PSYCHOSIS, ANXIETY DISORDERS, PANIC DISORDER, OBSESSIVE COMPULSIVE DISORDER, DEPRESSION, IMPULSE CONTROL DISORDERS, ALCOHOL ABUSE, AGGRESSION H. LUNDBECK A/S (DK) 1999-10-26 US disclosed
US-5807889-A PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS H. LUNDBECK A/S (DK) 1998-09-15 US disclosed
EP-0673360-B1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES LUNDBECK & CO AS H (DK) 1998-08-26 EP disclosed
EP-0673360-A1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES H. LUNDBECK A/S (DK) 1995-09-27 EP disclosed
WO-1994013620-A1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES H. LUNDBECK A/S (DK) 1994-06-23 WO disclosed