SCHEMBL8436852

SCHEMBL8436852

CC1CCc2ccc(NC=O)cc21.CCCNCCC

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.38
OPRD1 P41143 3/20 0.37
ACHE P22303 3/20 0.36
ADRA2A P08913 1/20 0.35
DRD2 P14416 2/20 0.33
DRD3 P35462 2/20 0.33
HTR1A P08908 1/20 0.33
DRD4 P21917 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
NQO2 P16083 2/20 0.33
MTNR1B P49286 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL8432169 0.94 MTNR1A (0.39) MTNR1AOPRD1ACHEDRD2DRD3
Dimethylamine SCHEMBL8433452 0.88 OPRD1 (0.38) MTNR1AOPRD1ADRA2AHTR1A
SCHEMBL8697680 0.84 MTNR1A (0.36) MTNR1AOPRD1ACHEADRA2ADRD2
SCHEMBL8435308 0.83 ADRA2A (0.43) MTNR1AADRA2ADRD2HTR1A
SCHEMBL8433416 0.82 MTNR1A (0.58) MTNR1AACHEADRA2AHTR1A
SCHEMBL8436872 0.80 MTNR1A (0.45) MTNR1AOPRD1ACHEDRD2
SCHEMBL8432637 0.79 MTNR1A (0.44) MTNR1AACHEDRD2DRD3HTR1A
SCHEMBL9627831 0.78 DRD2 (0.51) MTNR1ADRD2DRD3HTR1ADRD4
SCHEMBL8435260 0.78 ACHE (0.38) MTNR1AACHEDRD2DRD3HTR1A
SCHEMBL8432113 0.77 NPC1 (0.49) MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972964-A FOR TREATMENT OF CERTAIN PSYCHIC AND NEUROLOGIC DISORDERS SUCH AS PSYCHOSIS, ANXIETY DISORDERS, PANIC DISORDER, OBSESSIVE COMPULSIVE DISORDER, DEPRESSION, IMPULSE CONTROL DISORDERS, ALCOHOL ABUSE, AGGRESSION H. LUNDBECK A/S (DK) 1999-10-26 US disclosed
US-5807889-A PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS H. LUNDBECK A/S (DK) 1998-09-15 US disclosed
EP-0673360-B1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES LUNDBECK & CO AS H (DK) 1998-08-26 EP disclosed
EP-0673360-A1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES H. LUNDBECK A/S (DK) 1995-09-27 EP disclosed
WO-1994013620-A1 AMINOMETHYLINDANS, -BENZOFURANES AND -BENZOTHIOPHENES H. LUNDBECK A/S (DK) 1994-06-23 WO disclosed