SCHEMBL8437211

SCHEMBL8437211

COc1ccc2c3c(ccc2c1)C(C)(C)CCC3=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.41
ALDH1A1 P00352 3/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
CYP3A4 P08684 1/20 0.39
THRB P10828 1/20 0.39
MAPK1 P28482 1/20 0.39
GSTP1 P09211 1/20 0.38
ALOX5 P09917 1/20 0.38
MTNR1A P48039 3/20 0.37
MTNR1B P49286 3/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 2/20 0.37
TP53 P04637 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CYP2A6 P11509 2/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713153 0.78 GSTP1 (0.43) HSP90AA1ALDH1A1GRIN1GRIN2AGRIN2B
SCHEMBL31650634 0.77 KDM4E (0.45) ALDH1A1GRIN1GRIN2AGRIN2BCYP3A4
SCHEMBL2061344 0.77 KDM4E (0.45) ALDH1A1GRIN1GRIN2AGRIN2BCYP3A4
SCHEMBL1808153 0.74 KDM4E (0.49) ALDH1A1CYP3A4THRBMAPK1SMN1; SMN2
SCHEMBL31656371 0.70 MTNR1A (0.43) ALDH1A1MAPK1MTNR1AMTNR1BCYP1A2
SCHEMBL4523687 0.70 ALDH1A1 (0.37) ALDH1A1CYP3A4THRBMAPK1SMN1; SMN2
SCHEMBL1495858 0.70 KDM1A (0.53) ALDH1A1CYP3A4THRBMAPK1SMN1; SMN2
SCHEMBL886664 0.69 PDE7A (0.51) ALDH1A1GRIN1GRIN2AGRIN2BCYP3A4
SCHEMBL4420031 0.69 RXRA (0.53) ALDH1A1CYP3A4THRBMAPK1
SCHEMBL29462816 0.69 RXRA (0.53) ALDH1A1CYP3A4THRBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5945561-A ANTIINFLAMMATORY AGENT, RHEUMATIC DISORDERS, SKIN DISORDERS,ANTISCARRING AGENT BRISTOL-MYERS SQUIBB COMPANY (US) 1999-08-31 US disclosed
WO-1998049136-A1 RETINOID-LIKE COMPOUNDS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-11-05 WO disclosed