SCHEMBL8442576

SCHEMBL8442576

CC(=O)N(c1ccncc1)c1csc2cccnc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.36
CASP3 P42574 1/20 0.36
CASP7 P55210 1/20 0.36
CASP9 P55211 1/20 0.36
CASP6 P55212 1/20 0.36
CASP8 Q14790 1/20 0.36
IRAK4 Q9NWZ3 2/20 0.35
CDC7 O00311 1/20 0.34
PLK4 O00444 1/20 0.34
DAPK3 O43293 1/20 0.34
ROCK2 O75116 1/20 0.34
CHEK2 O96017 1/20 0.34
PIM1 P11309 1/20 0.34
FLT4 P35916 1/20 0.34
KDR P35968 1/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
RPS6KA3 P51812 1/20 0.34
PRKX P51817 1/20 0.34
PLK1 P53350 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9004605 0.86 IRAK4 (0.33) IRAK4CDC7LIMK1SMN1; SMN2L3MBTL1
SCHEMBL8440150 0.79 CHRM5 (0.36) IRAK4SMN1; SMN2L3MBTL1NPC1RAB9A
SCHEMBL8439945 0.79 LMNA (0.34) NSD2CASP3CASP7CASP9CASP6
SCHEMBL8442574 0.76 CYP2A6 (0.41) CDC7PLK4DAPK3ROCK2CHEK2
SCHEMBL8438852 0.76 CDC7 (0.36) CASP7CDC7PLK4DAPK3ROCK2
SCHEMBL8439457 0.74 SLC6A2 (0.35) ALDH1A1KMT2AHSD17B10
SCHEMBL8439939 0.72 SLC6A2 (0.35) L3MBTL1KDM4EALDH1A1KMT2A
SCHEMBL17023631 0.69 IRAK4 (0.49) CASP3IRAK4LIMK1SMN1; SMN2L3MBTL1
SCHEMBL7342232 0.68 GAA (0.38) SMN1; SMN2NPC1RAB9AKDM4EALDH1A1
SCHEMBL10861810 0.66 PKM (0.58) IRAK4SMN1; SMN2NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856335-A GLYCINE PARTIAL AGONISTS. HOECHST MARION ROUSSEL, INC. (US) 1999-01-05 US disclosed
US-5519032-A ANTIDEPRESSANTS, ANXIOLYTICS, ANTIEMETICS, ANTIPSYCHOTIC HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
EP-0581106-A1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-02-02 EP disclosed
US-5252581-A Modulators of neurotransmitters HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-10-12 US disclosed