SCHEMBL8438955

SCHEMBL8438955

O=C(c1cncnc1C1CC1)c1cccc(Cl)c1Cl

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.46
TSHR P16473 1/20 0.41
JAK2 O60674 1/20 0.38
PAK1 Q13153 2/20 0.37
ALOX12 P18054 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329113 0.75 RBP4 (0.44) TSHR
SCHEMBL8331089 0.73 ELANE (0.39)
SCHEMBL7032023 0.72 TSHR (0.71) P2RX7TSHRJAK2L3MBTL1TAS1R3
SCHEMBL9113731 0.72 P2RX7 (0.47) P2RX7TSHRALOX12L3MBTL1TAS1R3
SCHEMBL1014875 0.72 DHODH (0.38) L3MBTL1
SCHEMBL3823060 0.70 PARP1 (0.38)
SCHEMBL9134364 0.69 TSHR (0.65) P2RX7TSHRJAK2L3MBTL1TAS1R3
SCHEMBL8606571 0.68 TSHR (0.63) P2RX7TSHRJAK2L3MBTL1TAS1R3
SCHEMBL1015210 0.67 KDM4E (0.38) TSHRL3MBTL1
SCHEMBL534385 0.63 P2RX7 (1.00) P2RX7TSHRJAK2PAK1TAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939756-A2 A PROCESS FOR THE STEREOSELECTIVE REDUCTION OF ALPHA,BETA-UNSATURATED KETONES CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1999-09-08 EP disclosed
EP-0929510-A2 PROCESSES FOR THE PREPARATION OF ARYL-$g(b)-DIKETONES, ARYL-PYRIMIDINE KETONES AND CROP PROTECTION INTERMEDIATES ZENECA LIMITED (GB) 1999-07-21 EP disclosed
US-5925795-A Processes for the preparation of aryl-β-diketones, arylpyrimidine ketones and crop protection intermediates ZENECA LIMITED (GB) 1999-07-20 US disclosed
WO-1998011046-A2 PROCESSES FOR THE PREPARATION OF ARYL-β-DIKETONES, ARYL-PYRIMIDINE KETONES AND CROP PROTECTION INTERMEDIATES ZENECA LIMITED (GB) 1998-03-19 WO disclosed
WO-1997022602-A2 A PROCESS FOR THE STEREOSELECTIVE REDUCTION OF α,β-UNSATURATED KETONES CHINOIN, Gyógyszer és Vegyészeti (HU) 1997-06-26 WO disclosed