SCHEMBL8440710

SCHEMBL8440710

C=C1/C(=C\C=C2CCC[C@@]3(C)C2CC[C@@H]3[C@H](C)CCCC(C)C)C[C@@](O)(OO)C(O)(F)C1F

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 3/20 0.61
SLC6A2 P23975 2/20 0.61
AGTR1 P30556 2/20 0.61
VDR P11473 5/20 0.60
MAPT P10636 4/20 0.60
MEN1 O00255 3/20 0.60
KMT2A Q03164 3/20 0.60
CDC25A P30304 3/20 0.60
ALDH1A1 P00352 2/20 0.60
CYP3A4 P08684 2/20 0.60
ALOX15 P16050 2/20 0.60
PGR P06401 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
TDP1 Q9NUW8 1/20 0.60
HSPD1 P10809 1/20 0.60
HPGD P15428 1/20 0.60
TBXA2R P21731 1/20 0.60
PTGS1 P23219 1/20 0.60
GLRA1 P23415 1/20 0.60
DRD3 P35462 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4281111 0.87 VDR (0.68) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL11352175 0.82 MAPT (0.68) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL4974568 0.81 VDR (0.70) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL3698818 0.81 MAPT (0.69) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL260762 0.81 MAPT (0.69) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL6842113 0.81 MAPT (0.69) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL10034118 0.81 MAPT (0.69) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL9330205 0.81 MAPT (0.71) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL4979145 0.80 CDC25A (0.60) ADORA3SLC6A2AGTR1VDRMAPT
SCHEMBL10937380 0.80 ADORA3 (0.75) ADORA3SLC6A2AGTR1VDRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0833633-A4 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO INC (US) 1999-03-24 EP disclosed
EP-0833633-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1998-04-08 EP disclosed