SCHEMBL8440150

SCHEMBL8440150

CN(c1ccncc1)c1csc2cccnc12

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.36
CHKA P35790 1/20 0.36
NPC1 O15118 3/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
HSP90AA1 P07900 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPK14 Q16539 3/20 0.32
GRIA1 P42261 1/20 0.32
KDM4E B2RXH2 1/20 0.32
RAB9A P51151 1/20 0.32
PDE10A Q9Y233 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
GFER P55789 1/20 0.31
CYP19A1 P11511 1/20 0.30
ABCB1 P08183 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8439461 0.81 ALDH1A1 (0.34) CHRM5CHKANPC1L3MBTL1HSP90AA1
SCHEMBL8442576 0.79 NSD2 (0.36) NPC1L3MBTL1SMN1; SMN2KDM4ERAB9A
SCHEMBL8439457 0.79 SLC6A2 (0.35)
SCHEMBL8039461 0.78 MAPT (0.39) CHRM5CHKAMAPTSMN1; SMN2RAB9A
SCHEMBL8439939 0.77 SLC6A2 (0.35) L3MBTL1HSP90AA1MAPTKDM4E
Hydrochloric Acid SCHEMBL8039050 0.77 MAPT (0.38) CHRM5CHKAMAPTSMN1; SMN2RAB9A
SCHEMBL9004605 0.76 IRAK4 (0.33) NPC1L3MBTL1HSP90AA1SMN1; SMN2KDM4E
SCHEMBL8435363 0.76 CHKA (0.36) CHRM5CHKANPC1L3MBTL1HSP90AA1
SCHEMBL8440253 0.72 CHRM5 (0.38) CHRM5CHKANPC1MAPTSMN1; SMN2
SCHEMBL8440409 0.72 CYP2A6 (0.43) CHRM5CHKANPC1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856335-A GLYCINE PARTIAL AGONISTS. HOECHST MARION ROUSSEL, INC. (US) 1999-01-05 US disclosed
US-5519032-A ANTIDEPRESSANTS, ANXIOLYTICS, ANTIEMETICS, ANTIPSYCHOTIC HOECHST MARION ROUSSEL INC. (US) 1996-05-21 US disclosed
EP-0581106-A1 Substituted aminothienopyridines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-02-02 EP disclosed
US-5252581-A Modulators of neurotransmitters HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-10-12 US disclosed