SCHEMBL8443448

SCHEMBL8443448

CCCNC(C)c1ccc(Cl)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.48
HTR7 P34969 2/20 0.48
HTR6 P50406 2/20 0.48
CYP3A4 P08684 2/20 0.44
CHRM2 P08172 1/20 0.44
ADRA2A P08913 1/20 0.44
ADORA3 P0DMS8 1/20 0.44
CHRM1 P11229 1/20 0.44
SMPD1 P17405 1/20 0.44
DRD1 P21728 1/20 0.44
TBXA2R P21731 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
ADRA1A P35348 1/20 0.44
OPRM1 P35372 1/20 0.44
DRD3 P35462 1/20 0.44
CASR P41180 1/20 0.44
HTR2B P41595 1/20 0.44
SLC6A3 Q01959 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13975423 0.89 HTR1A (0.46) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL12849016 0.83 ADRB2 (0.46) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL12849094 0.83 ADRB2 (0.46) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL13074266 0.83 ADRB2 (0.46) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL172641 0.82 HTR1A (0.54) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL31579895 0.82 HTR1A (0.47) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL18687596 0.82 TAAR1 (0.47) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL13137645 0.82 SMN1; SMN2 (0.49) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL13911202 0.82 SMN1; SMN2 (0.49) HTR1AHTR7HTR6CYP3A4CHRM2
SCHEMBL13137652 0.81 ALDH1A1 (0.57) HTR1AHTR6CYP3A4SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0933354-B1 CALCIUM RECEPTOR-ACTIVE COMPOUNDS KYOWA HAKKO KIRIN CO LTD (JP) 2011-03-30 EP disclosed
EP-0618907-B1 1-(ARYLALKYL-AMINOALKYL)IMIDAZOLE DERIVATIVES, PROCESSES OF PREPARATION AND USE AS THERAPEUTICAL AGENTS BRITISH TECH GROUP INT (GB) 1999-04-28 EP disclosed
CN-1096781-A The therapeutical agent that contains 1-(aralkyl-aminoalkyl) imidazolium compounds BOOTS CO PLC (GB) 1994-12-28 CN disclosed