SCHEMBL8444573

SCHEMBL8444573

COc1cc(-c2nn(C)c(C(F)(F)F)c2Cl)c(F)cc1C#N

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 8/20 0.36
PGR P06401 1/20 0.36
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
EGFR P00533 3/20 0.33
KDM1A O60341 1/20 0.33
ERBB2 P04626 2/20 0.33
SCN9A Q15858 2/20 0.33
PDE2A O00408 1/20 0.32
PDE10A Q9Y233 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32
CHEK1 O14757 1/20 0.32
LRRK2 Q5S007 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7967445 0.87 TRPV4 (0.37) KDM1ASCN9AMEN1CYP1A2CYP2C9
SCHEMBL8440236 0.86 GPBAR1 (0.33) SCN9AMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL4625485 0.85 BCAT2 (0.44) ARSCN9A
SCHEMBL5398257 0.84 CYP1A2 (0.35) HSP90AA1HSP90AB1PDE2APDE10AMEN1
SCHEMBL7164579 0.83 MEN1 (0.33) ARMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8566825 0.82 GAA (0.36) EGFRSCN9APDE2APDE10AMEN1
SCHEMBL8566841 0.77 ALDH1A1 (0.35) MEN1CYP1A2CYP2C19KMT2A
SCHEMBL6911424 0.75 MEN1 (0.33) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL6912537 0.75 MEN1 (0.33) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL8569813 0.75 ALDH1A1 (0.35) MEN1CYP1A2CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0897383-A1 3-CYANOARYL PYRAZOLES AND THEIR USE AS HERBICIDES BAYER AG (DE) 1999-02-24 EP disclosed
WO-1997040018-A1 3-CYANOARYL PYRAZOLES AND THEIR USE AS HERBICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-10-30 WO disclosed