SCHEMBL8446993

SCHEMBL8446993

CS(=O)(=O)c1cc(C(=O)O)ccc1Oc1ccc(C(=O)CSC2=NCCN2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.55
CYP2D6 P10635 2/20 0.55
MAPT P10636 6/20 0.42
ALDH1A1 P00352 3/20 0.42
TDP1 Q9NUW8 1/20 0.42
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.38
GFER P55789 2/20 0.36
KMT2A Q03164 2/20 0.36
ADRA2A P08913 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
THRA P10827 1/20 0.35
THRB P10828 1/20 0.35
USP2 O75604 1/20 0.35
ALOX15 P16050 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8444221 0.86 CYP3A4 (0.44) CYP3A4CYP2D6MAPTALDH1A1TDP1
SCHEMBL8073894 0.81 CTSZ (0.45) MAPTALDH1A1GAAKMT2ATHRA
SCHEMBL8068695 0.80 ADRA1A (0.42) ADRA2AADRA1DADRA1AADRA1BTHRA
SCHEMBL8446994 0.80 RAB9A (0.53) MAPTALDH1A1LMNAKMT2ASMN1; SMN2
SCHEMBL8073502 0.76 TTR (0.51) MAPTALDH1A1GAATTR
SCHEMBL8446364 0.76 CA1 (0.55) MAPTALDH1A1GAAKMT2ASMN1; SMN2
SCHEMBL8068490 0.76 TTR (0.44) MAPTALDH1A1KMT2ASMN1; SMN2THRA
SCHEMBL11884885 0.72 CYP3A4 (1.00) CYP3A4CYP2D6MAPTALDH1A1TDP1
SCHEMBL7995261 0.72 TTR (0.61) ALDH1A1TDP1TTR
SCHEMBL8059681 0.72 TTR (0.45) MAPTGAAGFERSMN1; SMN2TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0723956-B1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AG (DE) 1999-10-13 EP disclosed
EP-0723956-A1 Basically substituted benzoylguanidines, process for their preparation, their use as medicaments or diagnostics as well as medicaments containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-07-31 EP disclosed