SCHEMBL8447229

SCHEMBL8447229

COC(=O)C(CCCN)NC(=O)OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 3/20 0.59
SIRT1 Q96EB6 3/20 0.59
SIRT3 Q9NTG7 3/20 0.59
PRSS1 P07477 2/20 0.59
PRSS2 P07478 2/20 0.59
PRSS3 P35030 2/20 0.59
TPSAB1 Q15661 2/20 0.59
KYNU Q16719 1/20 0.58
ALDH1A1 P00352 1/20 0.56
ALOX15 P16050 1/20 0.56
CTSL P07711 2/20 0.56
CTSS P25774 1/20 0.56
ITGB3 P05106 4/20 0.56
ITGA2B P08514 4/20 0.56
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
TLR2 O60603 1/20 0.52
CTSK P43235 2/20 0.52
DPP4 P27487 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8447232 1.00 SIRT2 (0.59) SIRT2SIRT1SIRT3PRSS1PRSS2
Hydrochloric Acid SCHEMBL6236103 0.99 SIRT2 (0.58) SIRT2SIRT1SIRT3PRSS1PRSS2
Hydrochloric Acid SCHEMBL6236109 0.99 SIRT2 (0.58) SIRT2SIRT1SIRT3PRSS1PRSS2
SCHEMBL6477219 0.96 SIRT2 (0.61) SIRT2SIRT1SIRT3PRSS1PRSS2
SCHEMBL1840309 0.96 SIRT2 (0.61) SIRT2SIRT1SIRT3PRSS1PRSS2
SCHEMBL1840311 0.96 SIRT2 (0.61) SIRT2SIRT1SIRT3PRSS1PRSS2
Hydrochloric Acid SCHEMBL6528872 0.95 SIRT2 (0.60) SIRT2SIRT1SIRT3PRSS1PRSS2
Hydrochloric Acid SCHEMBL3952159 0.95 SIRT2 (0.60) SIRT2SIRT1SIRT3PRSS1PRSS2
Hydrochloric Acid SCHEMBL3952162 0.95 SIRT2 (0.60) SIRT2SIRT1SIRT3PRSS1PRSS2
SCHEMBL22029461 0.92 KYNU (0.60) SIRT2SIRT1SIRT3KYNUALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0543997-B1 DERIVATIVES OF METHOTREXATE WITH ANTIRHEUMATIC ACTIVITY CHUGAI PHARMACEUTICAL CO LTD (JP) 1999-12-08 EP disclosed
EP-0543997-A1 NOVEL METHOTREXATE DERIVATIVE Chugai Seiyaku Kabushiki Kaisha (JP) 1993-06-02 EP disclosed