SCHEMBL8448979

SCHEMBL8448979

CN(C[C@@H]1CCN(C(=O)[C@@H]2C[C@H](S)CN2C)C1)C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 8/20 0.37
NR1D1 P20393 2/20 0.36
ALDH1A1 P00352 2/20 0.36
NR1H3 Q13133 1/20 0.36
NR1D2 Q14995 1/20 0.36
HTT P42858 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
ATM Q13315 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8447364 1.00 CCR5 (0.37) CCR5NR1D1ALDH1A1NR1H3NR1D2
SCHEMBL7450103 0.90 GRIN2B (0.37) CCR5NR1D1ALDH1A1NR1H3NR1D2
SCHEMBL8447213 0.90 GRIN2B (0.37) CCR5NR1D1ALDH1A1NR1H3NR1D2
SCHEMBL8444872 0.89 ALDH1A1 (0.35) CCR5NR1D1ALDH1A1NR1H3NR1D2
SCHEMBL8449100 0.89 ALDH1A1 (0.35) CCR5NR1D1ALDH1A1NR1H3NR1D2
SCHEMBL8447418 0.86 DPP8 (0.34) CCR5NR1D1ALDH1A1NR1H3NR1D2
SCHEMBL8447416 0.86 DPP8 (0.34) CCR5NR1D1ALDH1A1NR1H3NR1D2
SCHEMBL8448811 0.85 ALDH1A1 (0.34) CCR5NR1D1ALDH1A1NR1H3NR1D2
SCHEMBL8447420 0.85 NR1D1 (0.35) CCR5NR1D1NR1H3NR1D2ATM
SCHEMBL8449407 0.84 ALDH1A1 (0.38) CCR5ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977097-A 1-methylcarbapenem derivatives SANKYO COMPANY LIMITED (JP) 1999-11-02 US disclosed
EP-0900797-A1 1-METHYLCARBAPENEM DERIVATIVES SANKYO COMPANY LIMITED (JP) 1999-03-10 EP disclosed