SCHEMBL845441

SCHEMBL845441

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3CCCN3C(=O)Cc3ccccn3)cc2)cc1)[C@@H]1C=CCN1C(=O)Cc1ccccn1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.43
MAPK1 P28482 2/20 0.41
HCRTR1 O43613 2/20 0.41
HCRTR2 O43614 2/20 0.41
PABPC1 P11940 1/20 0.40
LMNA P02545 2/20 0.39
EPHX2 P34913 2/20 0.39
CYP3A4 P08684 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HTT P42858 1/20 0.37
ITGB1 P05556 2/20 0.37
ITGA4 P13612 2/20 0.37
TRPV1 Q8NER1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845195 0.91 HCRTR1 (0.46) GAAMAPK1HCRTR1HCRTR2PABPC1
SCHEMBL845190 0.91 EPHX2 (0.42) MAPK1EPHX2CYP3A4ITGB1ITGA4
SCHEMBL845393 0.89 GAA (0.47) GAAMAPK1HCRTR1HCRTR2PABPC1
SCHEMBL845086 0.88 EPHX2 (0.40) EPHX2CYP3A4ALDH1A1KDM4EITGB1
SCHEMBL845286 0.87 ALDH1A1 (0.48) GAAHCRTR1HCRTR2PABPC1LMNA
SCHEMBL845334 0.83 ITGB1 (0.39) EPHX2CYP3A4ITGB1ITGA4
SCHEMBL10119279 0.83 EPHX2 (0.37) MAPK1EPHX2CYP3A4ITGB1ITGA4
SCHEMBL10119337 0.77 ADRB1 (0.36) EPHX2CYP3A4ITGB1ITGA4
SCHEMBL15116912 0.77 ALDH1A1 (0.56) MAPK1HCRTR1HCRTR2PABPC1LMNA
SCHEMBL845205 0.77 ALDH1A1 (0.56) MAPK1HCRTR1HCRTR2PABPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed