SCHEMBL845334

SCHEMBL845334

O=C(Nc1ccc(/C=C/c2ccc(NC(=O)[C@@H]3C=CCN3C(=O)Cc3ccccn3)cc2)cc1)[C@@H]1C=CCN1C(=O)Cc1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.39
ITGA4 P13612 1/20 0.39
NAMPT P43490 1/20 0.39
PAX8 Q06710 1/20 0.38
CYP3A4 P08684 1/20 0.37
EPHX2 P34913 1/20 0.37
ADRB1 P08588 1/20 0.37
HRH3 Q9Y5N1 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA7 P36544 1/20 0.36
CHRNA4 P43681 1/20 0.36
POLB P06746 1/20 0.36
HTR1A P08908 1/20 0.35
DRD2 P14416 1/20 0.35
TBXAS1 P24557 1/20 0.35
MEN1 O00255 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
ROCK2 O75116 1/20 0.35
HDAC1 Q13547 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845622 0.92 ITGB1 (0.42) ITGB1ITGA4NAMPTPAX8HRH3
SCHEMBL845190 0.91 EPHX2 (0.42) ITGB1ITGA4CYP3A4EPHX2HTR1A
SCHEMBL10119337 0.89 ADRB1 (0.36) ITGB1ITGA4NAMPTPAX8CYP3A4
SCHEMBL845351 0.89 ITGB1 (0.41) ITGB1ITGA4NAMPTPAX8HRH3
SCHEMBL845086 0.88 EPHX2 (0.40) ITGB1ITGA4CYP3A4EPHX2HTR1A
SCHEMBL872288 0.84 ITGB1 (0.37) ITGB1ITGA4NAMPTPAX8HRH3
SCHEMBL10119279 0.83 EPHX2 (0.37) ITGB1ITGA4CYP3A4EPHX2HTR1A
SCHEMBL845441 0.83 GAA (0.43) ITGB1ITGA4CYP3A4EPHX2
SCHEMBL845099 0.81 ITGB1 (0.44) ITGB1ITGA4POLBHPGDKMT2A
SCHEMBL845098 0.77 ITGB1 (0.43) ITGB1ITGA4POLBHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed