SCHEMBL845570

SCHEMBL845570

CCc1ccnc(C(=O)N2CCC[C@H]2C(=O)Nc2ccc(/C=C/c3ccc(NC(=O)[C@@H]4CCCN4C(=O)c4cc(CC)ccn4)cc3)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53BP1 Q12888 1/20 0.45
KDM4E B2RXH2 2/20 0.44
LMNA P02545 1/20 0.44
PABPC1 P11940 1/20 0.43
ALDH1A1 P00352 2/20 0.43
RHOC P08134 1/20 0.42
RHOA P61586 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
CFTR P13569 3/20 0.42
GAA P10253 1/20 0.42
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAPK10 P53779 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL845685 0.93 TP53BP1 (0.46) TP53BP1KDM4ELMNAPABPC1ALDH1A1
SCHEMBL13272513 0.87 CFTR (0.38) TP53BP1KDM4ELMNAPABPC1ALDH1A1
SCHEMBL13272494 0.87 TP53BP1 (0.38) TP53BP1KDM4ELMNAPABPC1ALDH1A1
SCHEMBL845048 0.82 DGAT1 (0.50) KDM4ELMNAPABPC1ALDH1A1RHOC
SCHEMBL845405 0.82 TRPV1 (0.46) KDM4ERHOCRHOARXFP1CYP2C9
SCHEMBL845935 0.81 PABPC1 (0.44) TP53BP1KDM4ELMNAPABPC1ALDH1A1
SCHEMBL845250 0.78 HCRTR1 (0.46) TP53BP1KDM4ELMNAPABPC1ALDH1A1
SCHEMBL845333 0.78 PABPC1 (0.48) KDM4ELMNAPABPC1ALDH1A1RHOC
SCHEMBL845070 0.78 TRPV1 (0.44) KDM4ELMNAPABPC1ALDH1A1RHOC
SCHEMBL845007 0.77 PABPC1 (0.49) KDM4ELMNAPABPC1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed
US-8143288-B2 Inhibitors of HCV replication BRISTOL-MYERS SQUIBB COMPANY (US) 2012-03-27 US disclosed