SCHEMBL8458438

SCHEMBL8458438

N=C(N)NCCNC(=O)c1ccccc1C(=O)OC(=O)C[C@@H](N)NS(=O)(=O)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC1A3 P43003 2/20 0.36
SLC1A2 P43004 2/20 0.36
SLC1A1 P43005 2/20 0.36
KCNA5 P22460 1/20 0.36
PSMB8 P28062 4/20 0.35
PSMB5 P28074 4/20 0.35
USP2 O75604 1/20 0.35
ITGB3 P05106 5/20 0.35
ITGA2B P08514 4/20 0.35
CA9 Q16790 2/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA12 O43570 1/20 0.33
MMP2 P08253 1/20 0.33
CA14 Q9ULX7 1/20 0.33
KDM4E B2RXH2 2/20 0.33
ITGAV P06756 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7402176 0.88 USP2 (0.44) PSMB8PSMB5USP2ITGB3ITGA2B
SCHEMBL8801722 0.85 MMP1 (0.44) PSMB8PSMB5USP2ITGB3ITGA2B
SCHEMBL7487574 0.80 ITGB3 (0.48) ITGB3ITGA2BITGAVNPC1RAB9A
SCHEMBL7484657 0.79 ITGB3 (0.48) ITGB3ITGA2BCA9CA1CA2
SCHEMBL7912610 0.78 F2 (0.42) ITGB3ITGA2BCA2ITGAV
SCHEMBL7920933 0.77 ITGB3 (0.47) ITGB3ITGA2BCA9CA1CA2
SCHEMBL8458587 0.77 SLC1A3 (0.47) SLC1A3SLC1A2SLC1A1ITGB3ITGA2B
SCHEMBL8801713 0.76 SLC1A2 (0.55) SLC1A3SLC1A2SLC1A1
SCHEMBL7398408 0.76 ITGB3 (0.50) PSMB8PSMB5USP2ITGB3ITGA2B
SCHEMBL8456795 0.76 HSD17B10 (0.39) MMP2RAB9AGAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5929120-A Guainidino, formamidino, amino and related compounds for inhibiting osteoclast-mediated bone resorption MERCK & CO., INC. (US) 1999-07-27 US disclosed
US-5741796-A Pyridyl and naphthyridyl compounds for inhibiting osteoclast-mediated bone resorption MERCK & CO., INC. (US) 1998-04-21 US disclosed