SCHEMBL7402176

SCHEMBL7402176

N=C(N)NCCNC(=O)c1ccc(C(=O)OC(=O)C[C@@H](N)NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.44
ITGB3 P05106 12/20 0.43
ITGA2B P08514 11/20 0.43
ITGAV P06756 2/20 0.42
PSMB8 P28062 1/20 0.39
PSMB5 P28074 1/20 0.39
MAPT P10636 2/20 0.38
ALDH1A1 P00352 1/20 0.38
PRSS1 P07477 1/20 0.38
CTSG P08311 1/20 0.38
CTRB1 P17538 1/20 0.38
CMA1 P23946 1/20 0.38
CA2 P00918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801722 0.91 MMP1 (0.44) USP2ITGB3ITGA2BITGAVPSMB8
SCHEMBL7398408 0.89 ITGB3 (0.50) USP2ITGB3ITGA2BITGAVPSMB8
SCHEMBL8458438 0.88 SLC1A3 (0.36) USP2ITGB3ITGA2BITGAVPSMB8
SCHEMBL7487574 0.87 ITGB3 (0.48) ITGB3ITGA2BITGAVALDH1A1
SCHEMBL7484657 0.87 ITGB3 (0.48) ITGB3ITGA2BITGAVALDH1A1CA2
SCHEMBL7912610 0.86 F2 (0.42) ITGB3ITGA2BITGAVCA2
SCHEMBL8458587 0.84 SLC1A3 (0.47) ITGB3ITGA2BALDH1A1
SCHEMBL7398124 0.82 POLB (0.45) ITGB3ITGA2BMAPTALDH1A1CA2
SCHEMBL7920933 0.81 ITGB3 (0.47) ITGB3ITGA2BPRSS1CA2
SCHEMBL8455738 0.80 GAA (0.42) MAPTALDH1A1PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1994012181-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1994-06-09 WO claimed
US-5648368-A ANTICOAGULANTS MERCK & CO., INC. (US) 1997-07-15 US disclosed
WO-1994012181-A1 FIBRINOGEN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1994-06-09 WO disclosed