SCHEMBL8458979

SCHEMBL8458979

COc1ccc(-c2cc(O)ccc2C(=O)c2ccc(O)cc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.55
MAPT P10636 5/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
ALDH1A1 P00352 3/20 0.52
LMNA P02545 2/20 0.52
HPGD P15428 2/20 0.52
MAPK1 P28482 2/20 0.52
HTT P42858 2/20 0.52
CYP1A2 P05177 1/20 0.52
PGR P06401 1/20 0.52
CYP2D6 P10635 1/20 0.52
SLC6A2 P23975 1/20 0.52
PDE4A P27815 1/20 0.52
CYP2C19 P33261 1/20 0.52
HRH1 P35367 1/20 0.52
SLC6A3 Q01959 1/20 0.52
PDE4D Q08499 1/20 0.52
MEN1 O00255 1/20 0.52
PKM P14618 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7495907 1.00 NPC1 (0.55) NPC1MAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL8458268 0.98 NPC1 (0.56) NPC1MAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL8458977 0.94 NPC1 (0.59) NPC1MAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL8458703 0.94 NPC1 (0.59) NPC1MAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL8460808 0.93 ALDH1A1 (0.57) NPC1MAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL8339910 0.92 NPC1 (0.50) NPC1MAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL7502103 0.88 NPC1 (0.66) NPC1MAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL7503318 0.87 MMP2 (0.58) NPC1MAPTSMN1; SMN2ALDH1A1LMNA
SCHEMBL9681370 0.83 SMN1; SMN2 (0.64) NPC1MAPTSMN1; SMN2ALDH1A1HPGD
SCHEMBL30374771 0.81 HPGD (0.71) NPC1MAPTSMN1; SMN2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999025706-A1 2-ARYL-3-AROYLBENZO[B]THIOPHENES USEFUL FOR THE TREATMENT OF ESTROGEN DEPRIVATION SYNDROME ELI LILLY AND COMPANY (US) 1999-05-27 WO claimed
WO-1999025706-A1 2-ARYL-3-AROYLBENZO[B]THIOPHENES USEFUL FOR THE TREATMENT OF ESTROGEN DEPRIVATION SYNDROME ELI LILLY AND COMPANY (US) 1999-05-27 WO disclosed