SCHEMBL8459143

SCHEMBL8459143

NC(=O)C(Cl)CC(=O)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
ALDH1A1 P00352 4/20 0.50
MAPK1 P28482 2/20 0.50
GSK3B P49841 2/20 0.50
TRPA1 O75762 1/20 0.50
HIF1A Q16665 1/20 0.50
KMT2A Q03164 5/20 0.48
MAPT P10636 5/20 0.48
MEN1 O00255 4/20 0.48
TDP1 Q9NUW8 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
CYP3A4 P08684 2/20 0.48
HPGD P15428 2/20 0.48
KDM4E B2RXH2 2/20 0.48
ALOX15 P16050 1/20 0.48
CES1 P23141 1/20 0.48
NPC1 O15118 1/20 0.46
PTPN1 P18031 1/20 0.45
L3MBTL1 Q9Y468 7/20 0.45
POLB P06746 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5552472 0.84 TSHR (0.64) TSHRALDH1A1MAPK1GSK3BTRPA1
SCHEMBL8534214 0.82 TSHR (0.57) TSHRALDH1A1MAPK1GSK3BTRPA1
SCHEMBL2255355 0.79 TSHR (0.63) TSHRALDH1A1MAPK1GSK3BTRPA1
SCHEMBL5990135 0.78 TSHR (0.61) TSHRALDH1A1MAPK1GSK3BTRPA1
SCHEMBL28049900 0.77 L3MBTL1 (0.62) TSHRALDH1A1MAPK1GSK3BTRPA1
SCHEMBL29394053 0.76 CES2 (0.53) ALDH1A1POLBLMNANPSR1
SCHEMBL5158714 0.76 TSHR (0.59) TSHRALDH1A1MAPK1GSK3BTRPA1
SCHEMBL28481770 0.76 TSHR (0.59) TSHRALDH1A1MAPK1GSK3BTRPA1
SCHEMBL2598225 0.76 TSHR (0.59) TSHRALDH1A1MAPK1GSK3BTRPA1
SCHEMBL8898345 0.76 TSHR (0.59) TSHRALDH1A1MAPK1GSK3BTRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0914319-A1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LIMITED (JP) 1999-05-12 EP disclosed
WO-1997044329-A1 DIARYLALKYL CYCLIC DIAMINE DERIVATIVES AS CHEMOKINE RECEPTOR ANTAGONISTS TEIJIN LIMITED (JP) 1997-11-27 WO disclosed