SCHEMBL8459147

SCHEMBL8459147

COc1ccc([C@@](C)(C[C@H](O[Si](C)(C)C(C)(C)C)[C@H](CC2CCCCC2)NC(=O)OC(C)(C)C)C(=O)O)c(OC)c1OC

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 1/20 0.39
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
REN P00797 14/20 0.36
CACNA1B Q00975 3/20 0.35
PGC P20142 1/20 0.35
CYP3A4 P08684 1/20 0.34
CTSD P07339 1/20 0.34
CTSE P14091 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8458003 0.86 REN (0.42) AAK1CTSSCTSKRENCACNA1B
SCHEMBL8462263 0.84 KLK5 (0.41) CTSSCTSK
SCHEMBL8459146 0.81 REN (0.40) AAK1CTSSCTSKRENCYP3A4
SCHEMBL8852989 0.81 REN (0.40) AAK1CTSSCTSKRENCYP3A4
SCHEMBL10777312 0.74 CTSS (0.46) AAK1CTSSCTSKRENCYP3A4
SCHEMBL7274874 0.74 CTSS (0.46) AAK1CTSSCTSKRENCYP3A4
SCHEMBL10772696 0.73 ATM (0.49) RENCYP3A4
SCHEMBL8458897 0.73 REN (0.45) RENCACNA1B
SCHEMBL8853149 0.73 REN (0.45) RENCACNA1B
SCHEMBL10777836 0.73 CTSS (0.44) AAK1CTSSCTSKRENCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5935976-A Antiviral ethers of aspartate protease substrate isosteres NOVARTIS CORPORATION (US) 1999-08-10 US disclosed