SCHEMBL8459308

SCHEMBL8459308

C=CC(=O)Nc1ccc(C(=C(CC)c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 3/20 0.57
PTGS2 P35354 2/20 0.57
ESR1 P03372 11/20 0.53
ESR2 Q92731 7/20 0.53
PGR P06401 2/20 0.53
CYP19A1 P11511 1/20 0.53
ALDH1A1 P00352 1/20 0.49
HPGD P15428 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29684447 0.85 TGM2 (0.72) TGM2CYP19A1ALDH1A1RAB9A
SCHEMBL13586721 0.80 TGM2 (0.64) TGM2CYP19A1ALDH1A1RAB9A
SCHEMBL8456134 0.79 ACACB (0.49) PTGS2ESR1ESR2PGRCYP19A1
SCHEMBL39036 0.79 TGM2 (0.72) TGM2ALDH1A1HPGDRAB9A
SCHEMBL10773604 0.76 PTGS2 (0.60) PTGS2ESR1ESR2PGRCYP19A1
SCHEMBL81209 0.75 TGM2 (1.00) TGM2
SCHEMBL641477 0.74 ESR1 (0.80) PTGS2ESR1ESR2PGRCYP19A1
Diethylamine SCHEMBL1262240 0.74 TGM2 (0.76) TGM2ALDH1A1
SCHEMBL7238545 0.74 ESR1 (0.68) PTGS2ESR1ESR2PGRCYP19A1
SCHEMBL7238542 0.74 ESR1 (0.68) PTGS2ESR1ESR2PGRCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5681835-A USEFUL FOR TREATING OSTEOPOROSIS GLAXO WELLCOME INC. (US) 1997-10-28 US claimed
US-5877219-A Non-steroidal ligands for the estrogen receptor GLAXO WELLCOMEINC. (US) 1999-03-02 US disclosed
US-5681835-A USEFUL FOR TREATING OSTEOPOROSIS GLAXO WELLCOME INC. (US) 1997-10-28 US disclosed