SCHEMBL8459765

SCHEMBL8459765

COC(=O)C(Br)c1ccc(O)c(Br)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 2/20 0.50
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
ESR1 P03372 2/20 0.40
LMNA P02545 1/20 0.40
MT-CO2 P00403 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP19A1 P11511 1/20 0.38
ESR2 Q92731 1/20 0.37
BLM P54132 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TSHR P16473 1/20 0.37
MET P08581 1/20 0.37
MKNK2 Q9HBH9 1/20 0.37
NR3C1 P04150 2/20 0.36
PGR P06401 1/20 0.36
AR P10275 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31614294 0.83 MT-CO2 (0.55) FOLH1KMT2AMEN1GAAESR1
SCHEMBL27640937 0.83 MT-CO2 (0.55) FOLH1KMT2AMEN1GAAESR1
SCHEMBL18890086 0.82 LMNA (0.41) FOLH1KMT2AMEN1LMNANPSR1
SCHEMBL7069500 0.80 FOLH1 (0.50) FOLH1KMT2AMEN1GAAESR1
SCHEMBL29234606 0.79 KIF11 (0.38) FOLH1KMT2AMEN1ESR1ESR2
SCHEMBL27965732 0.78 FOLH1 (0.49) FOLH1KMT2AMEN1NR3C1PGR
SCHEMBL1564938 0.77 CYP1A2 (0.50) KMT2AMEN1LMNANPSR1
SCHEMBL8881032 0.77 ESR1 (0.54) KMT2AESR1LMNAALOX15ESR2
SCHEMBL12607235 0.76 TSHR (0.45) KMT2AMEN1GAAESR1LMNA
SCHEMBL30523061 0.75 KMT2A (0.46) KMT2AMEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0906315-A1 SPIRO-PIPERIDINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 1999-04-07 EP disclosed
WO-1997049710-A1 SPIRO-PIPERIDINE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 1997-12-31 WO disclosed