SCHEMBL8465273

SCHEMBL8465273

Cc1ccn2c3c(nc2c1)-c1ccccc1C(=O)C3=O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.52
HSP90AB1 P08238 1/20 0.52
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
MAPT P10636 3/20 0.45
GAA P10253 2/20 0.45
CGAS Q8N884 1/20 0.45
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
PARP1 P09874 1/20 0.44
PKM P14618 1/20 0.44
NPC1 O15118 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
AKT1 P31749 1/20 0.43
AKT2 P31751 1/20 0.43
TP53 P04637 1/20 0.42
POLB P06746 1/20 0.42
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8465600 0.83 HSP90AA1 (0.52) HSP90AA1HSP90AB1ALDH1A1MAPTRAB9A
SCHEMBL8465085 0.81 HSP90AA1 (0.57) HSP90AA1HSP90AB1
SCHEMBL8465304 0.81 HSP90AA1 (0.61) HSP90AA1HSP90AB1
SCHEMBL8465216 0.80 HSP90AA1 (0.79) HSP90AA1HSP90AB1
SCHEMBL8465101 0.78 HSP90AA1 (0.50) HSP90AA1HSP90AB1KDM4EALDH1A1MAPT
SCHEMBL31237237 0.78 HSP90AA1 (0.50) HSP90AA1HSP90AB1KDM4EALDH1A1MAPT
Sulfuric Acid SCHEMBL8465210 0.74 HSP90AA1 (0.46) HSP90AA1HSP90AB1KDM4EALDH1A1MAPT
SCHEMBL13325930 0.73 AKT2 (0.69) KDM4EALDH1A1MAPTGAACGAS
SCHEMBL8464947 0.72 KDM4E (0.48) HSP90AA1HSP90AB1KDM4EALDH1A1MAPT
SCHEMBL8464965 0.72 HSP90AA1 (0.74) HSP90AA1HSP90AB1ALDH1A1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5981544-A Mono-- or diketone tetracyclic derivatives and therapeutical uses thereof LABORATOIRE INNOTHERA (FR) 1999-11-09 US claimed
US-5981544-A Mono-- or diketone tetracyclic derivatives and therapeutical uses thereof LABORATOIRE INNOTHERA (FR) 1999-11-09 US disclosed