SCHEMBL8465600

SCHEMBL8465600

O=C1C(=O)c2c(nc3cc(Cl)ccn23)-c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.52
HSP90AB1 P08238 1/20 0.52
PARP1 P09874 1/20 0.44
AKT1 P31749 1/20 0.43
AKT2 P31751 1/20 0.43
S100A4 P26447 1/20 0.42
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
AHR P35869 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MAOB P27338 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8465273 0.83 HSP90AA1 (0.52) HSP90AA1HSP90AB1PARP1AKT1AKT2
SCHEMBL8465216 0.80 HSP90AA1 (0.79) HSP90AA1HSP90AB1
SCHEMBL8468193 0.79 HSP90AA1 (0.51) HSP90AA1HSP90AB1PARP1AKT1AKT2
SCHEMBL8464823 0.78 S100A4 (0.42) HSP90AA1HSP90AB1S100A4IDO1TDO2
SCHEMBL8465447 0.72 HSP90AA1 (0.47) HSP90AA1HSP90AB1AKT1AKT2IDO1
SCHEMBL8465227 0.71 HSP90AA1 (0.63) HSP90AA1HSP90AB1PARP1AKT1AKT2
SCHEMBL8466530 0.70 HSP90AA1 (0.50) HSP90AA1HSP90AB1AKT1AKT2IDO1
SCHEMBL31237237 0.70 HSP90AA1 (0.50) HSP90AA1HSP90AB1PARP1AKT1AKT2
SCHEMBL8465416 0.70 HSP90AA1 (0.50) HSP90AA1HSP90AB1PARP1AKT1AKT2
SCHEMBL8465101 0.70 HSP90AA1 (0.50) HSP90AA1HSP90AB1PARP1AKT1AKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5981544-A Mono-- or diketone tetracyclic derivatives and therapeutical uses thereof LABORATOIRE INNOTHERA (FR) 1999-11-09 US claimed
US-5981544-A Mono-- or diketone tetracyclic derivatives and therapeutical uses thereof LABORATOIRE INNOTHERA (FR) 1999-11-09 US disclosed