SCHEMBL8465400

SCHEMBL8465400

CSC(=O)CC(=O)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FAAH O00519 12/20 0.43
CES1 P23141 10/20 0.42
CES2 O00748 6/20 0.41
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PLA2G6 O60733 1/20 0.39
PLOD2 O00469 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9065118 0.91 FAAH (0.38) FAAHCES1CES2MEN1CYP1A2
SCHEMBL615589 0.76 FAAH (0.45) FAAHCES1CES2MEN1CYP1A2
SCHEMBL183178 0.74 PLOD2 (0.46) FAAHCES1CES2MEN1CYP1A2
SCHEMBL12582310 0.74
SCHEMBL6517983 0.72 PLOD2 (0.44) FAAHCES1CES2MEN1CYP1A2
SCHEMBL9326020 0.72 PLOD2 (0.44) FAAHCES1CES2MEN1CYP1A2
SCHEMBL9283764 0.72 PLOD2 (0.44) FAAHCES1CES2MEN1CYP1A2
SCHEMBL6520648 0.72 PLOD2 (0.44) FAAHCES1CES2MEN1CYP1A2
Water SCHEMBL7191917 0.72 PLOD2 (0.44) FAAHCES1CES2MEN1CYP1A2
Water SCHEMBL7197275 0.72 PLOD2 (0.44) FAAHCES1CES2MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877210-A CONTROLLING IMMUNE RESPONSE BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-02 US claimed
US-5583242-A VANADYL COMPLEXES BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US claimed
US-5565491-A FOR TREATMENT OF DISEASES MARKED BY MALIGNANT PROLIFERATION OF B CELLS, SUCH AS LEUKEMIA AND LYMPHOMAS; ANTICARCINOGENIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1996-10-15 US claimed
EP-0448544-B1 Process for preparation of fluoromethyl-substituted piperidine carbodithioates ROHM & HAAS (US) 1996-07-03 EP claimed
EP-0448544-A2 Process for preparation of fluoromethyl-substituted piperidine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP claimed
US-4785129-A Methyl 4,4,4-trifluoro-3-oxo-butanethioate MONSANTO COMPANY (US) 1988-11-15 US claimed
US-20230241078-A1 Vanadyl and vanadate for use in reducing stress-induced metabolic derangement CFM PHARMA HOLDING B.V. (NL) 2023-08-03 US disclosed
US-20200246352-A1 Vanadyl and vanadate for use in reducing stress-induced metabolic derangement CFM PHARMA HOLDING B.V. (NL) 2020-08-06 US disclosed
EP-3412654-A1 PROCESSES FOR THE MANUFACTURE OF HALOALKYL PYRIMIDYL COMPOUNDS, AND COMPOUNDS USEFUL IN THEIR MANUFACTURE SOLVAY SA (BE) 2018-12-12 EP disclosed
US-5877210-A CONTROLLING IMMUNE RESPONSE BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-02 US disclosed
US-5846998-A Use of phosphotyrosine phosphatase inhibitors or phosphotyrosine kinase activators for controlling cellular proliferation BRISTOL-MYERS SQUIBB COMPANY (US) 1998-12-08 US disclosed
US-5693627-A TREATING DISEASES SUCH AS LEUKEMIAS AND LYMPHOMAS BRISTOL-MYERS SQUIBB COMPANY (US) 1997-12-02 US disclosed
US-5583242-A VANADYL COMPLEXES BRISTOL-MYERS SQUIBB COMPANY (US) 1996-12-10 US disclosed
EP-0448541-A2 Process for preparation of fluoromethyl-substituted pyridine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP disclosed
EP-0448543-A2 Process for preparation of fluoromethyl-substituted pyridine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP disclosed
EP-0448544-A2 Process for preparation of fluoromethyl-substituted piperidine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP disclosed
EP-0448542-A2 Process for preparation of fluoromethyl-substituted dihydropyridine carbodithioates ROHM AND HAAS COMPANY (US) 1991-09-25 EP disclosed
US-5051512-A Reaction of trifluoroacetic acid thiomethyl ester and ammonia, reaction with an alkyl aldehyde and heating MONSANTO COMPANY (US) 1991-09-24 US disclosed
US-4785129-A Methyl 4,4,4-trifluoro-3-oxo-butanethioate MONSANTO COMPANY (US) 1988-11-15 US disclosed
US-4785129-A Methyl 4,4,4-trifluoro-3-oxo-butanethioate MONSANTO COMPANY (US) 1988-11-15 US disclosed