SCHEMBL8468924

SCHEMBL8468924

O=C1N=Nc2nc[nH]c(=O)c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
PARP1 P09874 8/20 0.35
PDPK1 O15530 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CA12 O43570 1/20 0.35
ALOX15 P16050 1/20 0.35
CA9 Q16790 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
ADORA2A P29274 1/20 0.34
SLC6A4 P31645 1/20 0.34
ADRA1A P35348 1/20 0.34
XDH P47989 1/20 0.34
RAB9A P51151 1/20 0.34
BLM P54132 1/20 0.34
HPGD P15428 1/20 0.33
KDM4A O75164 1/20 0.32
KDM4B O94953 1/20 0.32
KDM5C P41229 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28672687 0.61 ALDH1A1 (0.41) ALDH1A1PARP1PDPK1SMN1; SMN2CA12
SCHEMBL4455591 0.61
SCHEMBL10612254 0.60 ALDH1A1 (0.31) ALDH1A1
SCHEMBL355917 0.60 ALDH1A1 (0.40) ALDH1A1PARP1PDPK1SMN1; SMN2CA12
SCHEMBL1867923 0.60 ALDH1A1 (0.40) ALDH1A1PARP1PDPK1SMN1; SMN2CA12
SCHEMBL5165263 0.59 ALDH1A1 (0.44) ALDH1A1BLMMAPK9MAPK14
Hypoxanthine SCHEMBL25381 0.59 ALDH1A1 (1.00) ALDH1A1PDPK1SMN1; SMN2LMNATSHR
Hypoxanthine SCHEMBL7037918 0.59 ALDH1A1 (1.00) ALDH1A1PDPK1SMN1; SMN2LMNATSHR
Hypoxanthine SCHEMBL30096461 0.59 ALDH1A1 (1.00) ALDH1A1PDPK1SMN1; SMN2LMNATSHR
SCHEMBL4781198 0.58 ALDH1A1 (0.39) ALDH1A1PARP1PDPK1SMN1; SMN2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496617-B1 Adenosine kinase inhibitors METABASIS THERAPEUTICS INC (US) 1999-12-01 EP disclosed
EP-0682519-A4 ADENOSINE KINASE INHIBITORS. GENSIA INC (US) 1997-12-17 EP disclosed
US-5646128-A TREATING INFLAMMATION, SEPSIS, SEPTIC SHOCK, BURNS GENSIA, INC. (US) 1997-07-08 US disclosed
EP-0682519-A1 ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1995-11-22 EP disclosed
WO-1994017803-A9 ADENOSINE KINASE INHIBITORS 1994-09-29 WO disclosed
WO-1994017803-A1 ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1994-08-18 WO disclosed
WO-1992012718-A1 ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1992-08-06 WO disclosed
EP-0496617-A1 Adenosine kinase inhibitors GENSIA, INC. (US) 1992-07-29 EP disclosed