SCHEMBL8469854

SCHEMBL8469854

O=C1NC(=O)c2c(CCCN3CCC(c4noc5cc(F)ccc45)CC3)cccc21

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.57
DRD2 P14416 5/20 0.56
SLC6A4 P31645 1/20 0.56
HTR2A P28223 3/20 0.56
HTR1A P08908 1/20 0.54
MCHR1 Q99705 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664537 0.97 DRD2 (0.57) ACHEDRD2SLC6A4HTR2A
SCHEMBL1545276 0.95 ACHE (0.59) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL7744954 0.84 DRD2 (0.52) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL1545853 0.83 ACHE (0.60) ACHEDRD2SLC6A4HTR2AHTR1A
Hydrochloric Acid SCHEMBL8627510 0.82 ACHE (0.56) ACHEDRD2SLC6A4HTR2A
SCHEMBL8788161 0.80 DRD2 (0.40) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL6644402 0.80 PARP1 (0.49) DRD2SLC6A4HTR2AHTR1A
SCHEMBL793140 0.78 DRD2 (0.70) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL791048 0.78 DRD2 (0.70) ACHEDRD2SLC6A4HTR2AHTR1A
SCHEMBL28972648 0.78 DRD2 (0.60) ACHEDRD2SLC6A4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889035-A 1-(Arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-3-(heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics HOECHST MARION ROUSSEL, INC. (US) 1999-03-30 US disclosed
US-5874435-A PSYCHOLOGICAL DISORDERS; ANALGESICS HOECHST MARION ROUSSEL, INC. (US) 1999-02-23 US disclosed
US-5854243-A 3-heteroaryl-1-pyrrolidinealkylthiols and derivatives thereof and their therapeutic utility HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1998-12-29 US disclosed
US-5843977-A (3-heteroaryl-1-pyrrolidinyl) alkoxy!-3,4-dihydro-1(2H)-naphthalenones and related compounds and their therapeutic utility HOECHST MARION ROSUEEL, INC. 1998-12-01 US disclosed
US-5840727-A ANTIPSYCHOTICS, ANALGESICS AVENTIS PHARMACEUTICALS INC. 1998-11-24 US disclosed
US-5811435-A 2- (4-heteroaryl-1-piperidinyl)alkyl!-1,3-dioxanes and related compounds and their therapeutic utility HOECHST MARION RUSSEL, INC. 1998-09-22 US disclosed