SCHEMBL8470221

SCHEMBL8470221

Cc1nc(-c2n[nH]c3cccc(Cc4ccccc4F)c23)oc1CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 1/20 0.34
ALDH1A1 P00352 3/20 0.34
ALDH3A1 P30838 1/20 0.34
PTDSS1 P48651 1/20 0.34
MAPT P10636 3/20 0.33
KMT2A Q03164 2/20 0.33
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 2/20 0.33
NPC1 O15118 2/20 0.33
MEN1 O00255 1/20 0.33
CDC7 O00311 1/20 0.33
PLK4 O00444 1/20 0.33
CHEK1 O14757 1/20 0.33
IKBKB O14920 1/20 0.33
RGS12 O14924 1/20 0.33
AURKA O14965 1/20 0.33
GAK O14976 1/20 0.33
PDPK1 O15530 1/20 0.33
DAPK3 O43293 1/20 0.33
DYRK3 O43781 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5312666 0.83 MAP4K1 (0.35) MAP4K1ALDH1A1KDM4EHSD17B10LMNA
SCHEMBL5314312 0.81 PPARD (0.34) MAP4K1MAPK1NPSR1PKM
SCHEMBL5419366 0.74 AR (0.32) MAP4K1ALDH1A1KDM4EJAK1MAPK1
SCHEMBL4425835 0.73 CHRM1 (0.44)
SCHEMBL5313810 0.71 MAP2K4 (0.37) KMT2ANPC1MEN1CYP1A2POLB
SCHEMBL5314525 0.69 MAPK1 (0.34) LMNACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4435380 0.69 MAPT (0.49) ALDH1A1MAPTKMT2AKDM4EHSD17B10
SCHEMBL5313829 0.68 ALDH1A1 (0.36) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8327060 0.66 AR (0.35) ALDH1A1MAPTKMT2AKDM4EHSD17B10
SCHEMBL7810926 0.65 AR (0.39) ALDH1A1KDM4ENPC1POLBMKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934311-A2 NEW HETEROCYCLYLMETHYL-SUBSTITUTED PYRAZOL DERIVATES BAYER AG (DE) 1999-08-11 EP disclosed
WO-1998016507-A2 NEW HETEROCYCLYLMETHYL-SUBSTITUTED PYRAZOL DERIVATES AND THEIR USE FOR TREATING CARDIOVASCULAR DISEASES BAYER AKTIENGESELLSCHAFT (DE) 1998-04-23 WO disclosed