SCHEMBL8474155

SCHEMBL8474155

[CH2]CC(=O)OCc1cccc2c1Cc1ccccc1-2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.51
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
HTR7 P34969 2/20 0.40
HTR2B P41595 2/20 0.40
DRD2 P14416 3/20 0.39
DRD4 P21917 2/20 0.39
DRD3 P35462 2/20 0.39
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34
GABRG2 P18507 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4059189 0.89 PNMT (0.54) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL5497718 0.87 PNMT (0.53) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL4839271 0.86 PNMT (0.51) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL8473288 0.86 PNMT (0.54) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL1830397 0.85 PNMT (0.57) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL6849876 0.85 PNMT (0.50) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL4059193 0.85 PNMT (0.50) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL8671794 0.84 PNMT (0.55) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL1830400 0.84 PNMT (0.55) PNMTNPC1RAB9AHTR7HTR2B
SCHEMBL19384366 0.84 RAB9A (0.50) PNMTNPC1RAB9AHTR7HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5859190-A SOLID PHASE SYNTHESIS TO FORM A PROTECTED DIPEPTIDE FOLLOWED BY REACTING WITH 1,1'-THIOCARBONYLDIIMIDAZOLE TO EFFECT RING FORMATION; EFFICIENCY; ANTICONVULSANT,-ARRHYTHMIC AND DIABETIC AGENTS; HERBICIDES AND FUNGICIDES TREGA BIOSCIENCES, INC. (US) 1999-01-12 US claimed
WO-1998033776-A1 COMBINATORIAL LIBRARIES OF HYDANTOIN AND THIOHYDANTOIN DERIVATIVES, METHODS OF MAKING THE LIBRARIES AND COMPOUNDS THEREIN TREGA BIOSCIENCES, INC. (US) 1998-08-06 WO claimed
US-5859190-A SOLID PHASE SYNTHESIS TO FORM A PROTECTED DIPEPTIDE FOLLOWED BY REACTING WITH 1,1'-THIOCARBONYLDIIMIDAZOLE TO EFFECT RING FORMATION; EFFICIENCY; ANTICONVULSANT,-ARRHYTHMIC AND DIABETIC AGENTS; HERBICIDES AND FUNGICIDES TREGA BIOSCIENCES, INC. (US) 1999-01-12 US disclosed
WO-1998033776-A1 COMBINATORIAL LIBRARIES OF HYDANTOIN AND THIOHYDANTOIN DERIVATIVES, METHODS OF MAKING THE LIBRARIES AND COMPOUNDS THEREIN TREGA BIOSCIENCES, INC. (US) 1998-08-06 WO disclosed