SCHEMBL8476147

SCHEMBL8476147

O=C(NC1CCCCCCC1)c1c(C(c2ccccc2)c2ccccc2)c2ccccc2n1CCCN1CCCC1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
CYP3A4 P08684 2/20 0.49
CYP2D6 P10635 2/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
CNR2 P34972 6/20 0.45
CNR1 P21554 3/20 0.45
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
KDM4E B2RXH2 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HTR4 Q13639 1/20 0.42
CCR5 P51681 1/20 0.42
LMNA P02545 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8477083 0.98 CYP3A4 (0.49) TSHRCYP3A4CYP2D6TP53CYP1A2
SCHEMBL8472493 0.87 KDM4E (0.52) TSHRCYP3A4CYP2D6TP53CYP1A2
SCHEMBL8472271 0.87 HRH3 (0.47) TP53CNR2CNR1KDM4ESMN1; SMN2
SCHEMBL8472267 0.86 KDM4E (0.45) TSHRCYP3A4CYP2D6CNR2CNR1
SCHEMBL8476064 0.85 KDM4E (0.44) TSHRCYP3A4CYP2D6CNR2CNR1
SCHEMBL8898545 0.84 CNR2 (0.44) TDP1CNR2KDM4ELMNA
SCHEMBL8475760 0.84 KDM4E (0.46) TSHRCYP3A4CYP2D6TP53CYP1A2
SCHEMBL8472179 0.84 KDM4E (0.48) TSHRCYP3A4CYP2D6TP53CYP1A2
SCHEMBL8473304 0.84 KDM4E (0.46) TSHRCYP3A4CYP2D6TP53CYP1A2
SCHEMBL8477838 0.84 CNR2 (0.48) CNR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5891902-A OSTEOPOROSIS KYOWA HAKKO KOGYO CO., LTD. (JP) 1999-04-06 US disclosed
EP-0782989-A1 INDOLE DERIVATIVES KYOWA HAKKO KOGYO CO., LTD. (JP) 1997-07-09 EP disclosed