SCHEMBL8476607

SCHEMBL8476607

CCc1noc(NS(=O)(=O)c2ccccc2)c1-c1ccc(C)cc1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 12/20 0.53
EDNRB P24530 10/20 0.53
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
HSD11B1 P28845 1/20 0.42
ALDH1A1 P00352 1/20 0.42
PKM P14618 1/20 0.42
MCL1 Q07820 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8479988 0.92 EDNRA (0.55) EDNRAEDNRBTSHRMAPK1ALDH1A1
SCHEMBL8481520 0.89 EDNRA (0.50) EDNRAEDNRBTSHRMAPK1HSD11B1
SCHEMBL8478164 0.86 HSD11B1 (0.49) EDNRAEDNRBHSD11B1
SCHEMBL8479975 0.85 EDNRA (0.66) EDNRAEDNRB
SCHEMBL8473239 0.82 EDNRA (0.52) EDNRAEDNRBTSHRMAPK1ALDH1A1
SCHEMBL9065130 0.82 EDNRA (0.69) EDNRAEDNRBTSHR
SCHEMBL7850015 0.82 EDNRA (0.69) EDNRAEDNRBTSHR
SCHEMBL8481482 0.81 TSHR (0.45) EDNRAEDNRBTSHRMAPK1CA12
SCHEMBL8523604 0.79 EDNRA (0.51) EDNRAEDNRBTSHRMAPK1
SCHEMBL8477061 0.79 EDNRA (0.50) EDNRAEDNRBTSHRMAPK1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5859257-A ANTIINFLAMMATORY, ANTIARTHRITIC AGENTS G. D. SEARLE & CO. (US) 1999-01-12 US disclosed