SCHEMBL8478069

SCHEMBL8478069

CCc1n[c]c(C)c(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HEXA P06865 3/20 0.44
HEXB P07686 3/20 0.44
DHFR P00374 1/20 0.44
GCGR P47871 2/20 0.40
PTGS1 P23219 2/20 0.38
PTGS2 P35354 2/20 0.38
TP53 P04637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
AKT2 P31751 2/20 0.34
BRD4 O60885 2/20 0.34
CHEK1 O14757 1/20 0.34
BRD2 P25440 1/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8474990 0.82 DHFR (0.44) HEXAHEXBDHFRGCGRPTGS1
SCHEMBL8474820 0.78 DHFR (0.41) HEXAHEXBDHFRGCGRPTGS1
SCHEMBL8475027 0.77 BRD4 (0.42) PTGS1PTGS2TP53L3MBTL1AKT2
SCHEMBL9076864 0.69 HEXA (0.53) HEXAHEXBDHFRGCGRPTGS1
SCHEMBL8479260 0.68 TP53 (0.41) HEXAHEXBDHFRGCGRPTGS1
SCHEMBL11720669 0.67 LMNA (0.43) PTGS1PTGS2L3MBTL1AKT2BRD4
SCHEMBL12368269 0.63 HEXA (0.73) HEXAHEXBDHFRTP53L3MBTL1
SCHEMBL8478772 0.62 BRD4 (0.36) DHFRGCGRTP53L3MBTL1AKT2
SCHEMBL31500058 0.62 ALDH1A1 (0.50) HEXAHEXBDHFRL3MBTL1KDM4E
SCHEMBL11738666 0.62 ADORA3 (0.49) HEXAHEXBDHFRPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6004988-A Carboxylic acid derivatives, their preparation and their use BASF AKTIENGESELLSCHAFT (DE) 1999-12-21 US disclosed