SCHEMBL8481123

SCHEMBL8481123

COC(=O)c1ccc(C(=O)c2c(F)cc(OC)cc2OC)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
KMT2A Q03164 6/20 0.52
NPC1 O15118 1/20 0.48
CYP3A4 P08684 2/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPT P10636 5/20 0.45
ALDH1A1 P00352 2/20 0.45
HTT P42858 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
GAA P10253 1/20 0.45
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
TAS1R2 Q8TE23 1/20 0.45
MEN1 O00255 3/20 0.44
KDM4E B2RXH2 1/20 0.44
TUBB4A P04350 1/20 0.44
TUBB P07437 1/20 0.44
TUBA3C P0DPH7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8128739 0.87 EGFR (0.46) CA1CA2KMT2ANPC1CYP3A4
SCHEMBL8481431 0.87 ALDH1A1 (0.56) CA1CA2KMT2ANPC1CYP3A4
SCHEMBL8480798 0.85 CA1 (0.53) CA1CA2KMT2ACYP3A4CYP2D6
SCHEMBL13963805 0.79 KMT2A (0.62) CA1CA2KMT2ACYP3A4CYP2D6
SCHEMBL8017091 0.77 CYP3A4 (0.55) CA1CA2CYP3A4ALDH1A1GAA
SCHEMBL3468486 0.77 LMNA (0.63) CA1CA2KMT2ANPC1CYP3A4
SCHEMBL18170324 0.76 MAPK1 (0.51) CA1CA2KMT2ACYP3A4CYP2D6
SCHEMBL18044458 0.76 CA1 (0.47) CA1CA2KMT2ANPC1CYP3A4
SCHEMBL21166953 0.75 CA1 (0.59) CA1CA2KMT2AMAPTALDH1A1
SCHEMBL4743101 0.75 HPGD (0.64) KMT2ANPC1MAPTNPSR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5914406-A ENZYME INHIBITOR; USEFUL FOR TREATMENT OF INFLAMMATORY SKIN DISORDERS AND ALOPECIA HOFFMAN-LA ROCHE INC. (US) 1999-06-22 US disclosed
US-5750706-A TREATMENT OF INFLAMMATORY SKIN DISORDERS AND ALOPECIA HOFFMANN-LA ROCHE INC. (US) 1998-05-12 US disclosed
US-5583222-A ANTIINFLAMMATORY AGENTS FOR TREATMENT OF SKIN DISORDERS HOFFMANN-LA ROCHE INC. (US) 1996-12-10 US disclosed