SCHEMBL848485

SCHEMBL848485

CC(=O)c1ccccc1Nc1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.68
ALOX15 P16050 1/20 0.68
MEN1 O00255 1/20 0.68
KMT2A Q03164 1/20 0.68
FABP4 P15090 1/20 0.67
AKR1C3 P42330 4/20 0.60
AKR1C2 P52895 4/20 0.60
SIRT2 Q8IXJ6 8/20 0.56
PTGS1 P23219 1/20 0.51
AKR1B10 O60218 1/20 0.51
AKR1B1 P15121 1/20 0.51
AKR1C4 P17516 1/20 0.51
AKR1C1 Q04828 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
MT-CO2 P00403 1/20 0.50
SIRT1 Q96EB6 1/20 0.50
POLB P06746 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30567367 1.00 MAPT (0.68) MAPTALOX15MEN1KMT2AFABP4
Acetonitrile SCHEMBL27301956 0.91 MEN1 (0.59) MAPTALOX15MEN1KMT2AFABP4
SCHEMBL25449209 0.87 AKR1C3 (0.66) MAPTALOX15MEN1KMT2AFABP4
SCHEMBL8052123 0.87 MEN1 (0.58) MAPTALOX15MEN1KMT2AFABP4
SCHEMBL10936401 0.87 MEN1 (0.58) MAPTALOX15MEN1KMT2AFABP4
Fenamic Acid SCHEMBL27925717 0.86 FABP4 (0.82) MAPTALOX15MEN1KMT2AFABP4
SCHEMBL30567365 0.85 MEN1 (0.56) MAPTALOX15MEN1KMT2AFABP4
SCHEMBL7844252 0.85 MEN1 (0.56) MAPTALOX15MEN1KMT2AFABP4
SCHEMBL6620978 0.85 AKR1C3 (0.57) MAPTALOX15MEN1KMT2AFABP4
SCHEMBL30982117 0.85 AKR1C3 (0.57) MAPTALOX15MEN1KMT2AFABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230381133-A1 TAU AND AMYLOID PROTEIN LOWERING COMPOUNDS AND METHODS OF USE HAMAD BIN KHALIFA UNIVERSITY (QA) 2023-11-30 US disclosed
CN-116589406-A Preparation method of polysubstituted acridine derivative 深圳职业技术学院 2023-08-15 CN disclosed
EP-3464317-B1 AMINOSTEROID DERIVATIVES AND PROCESS FOR PRODUCING SAME UNIV LAVAL (CA) 2023-04-26 EP disclosed
US-11174282-B2 Aminosteroid derivatives and process for producing same UNIVERSITé LAVAL (CA) 2021-11-16 US disclosed
WO-2017205964-A1 AMINOSTEROID DERIVATIVES AND PROCESS FOR PRODUCING SAME UNIVERSITé LAVAL (CA) 2017-12-07 WO disclosed
US-8653054-B2 2-(N-substituted piperazinyl) steroid derivatives UNIVERSITE LAVAL (CA) 2014-02-18 US disclosed
US-8653054-B2 2-(N-substituted piperazinyl) steroid derivatives UNIVERSITE LAVAL (CA) 2014-02-18 US disclosed
US-8163906-B2 Dihydroquinone and dihydronaphthridine inhibitors of JNK ROCHE PALO ALTO, LLC (US) 2012-04-24 US disclosed
EP-2148862-B1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK HOFFMANN LA ROCHE (CH) 2012-03-28 EP disclosed
US-20110312926-A1 2-(N-Substituted Piperazinyl) Steroid Derivatives UNIVERSITE LAVAL (CA) 2011-12-22 US disclosed
WO-2008138920-A1 DIHYDROQUINONE AND DIHYDRONAPHTHRIDINE INHIBITORS OF JNK F. HOFFMANN-LA ROCHE AG (CH) 2008-11-20 WO disclosed
US-7378154-B2 Radiation transparent glass, polycarbonate, polyethylene terephthalate, acrylic, methyl cellulose or polycycloolefin substrate, a fluoropolymer layer containing and a rare earth metal compound, and a low refractive index layer; fluorescence; light amplification; improved efficiency; light emitting diodes DAIKIN INDUSTRIES, LTD. (JP) 2008-05-27 US disclosed
EP-0783505-B1 PYRROLO[2,3-d]PYRIMIDINES AND THEIR USE NOVARTIS AG (CH) 2001-03-07 EP disclosed
CN-1046731-C Pyrrolo [2,3-d ] pyrimidines and their use NOVARTIS AG (CH) 1999-11-24 CN disclosed
US-5869485-A Pyrrolo 2,3-d!pyrimidines and their use NOVARTIS FINANCE CORP. (US) 1999-02-09 US disclosed
CN-1164234-A Pyrrolo [2, 3-d ] pyrimidines and their use NOVARTIS AG (CH) 1997-11-05 CN disclosed
EP-0783505-A1 PYRROLO[2,3-d]PYRIMIDINES AND THEIR USE Novartis AG (CH) 1997-07-16 EP disclosed
WO-1996010028-A1 PYRROLO[2,3-d]PYRIMIDINES AND THEIR USE NOVARTIS AG (CH) 1996-04-04 WO disclosed
US-5153226-A Administering as anticholesterol agents, for atherosclerosis WARNER-LAMBERT COMPANY (US) 1992-10-06 US disclosed
EP-0415413-A1 Acat inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230381133-A1 TAU AND AMYLOID PROTEIN LOWERING COMPOUNDS AND METHODS OF USE MAPT, TTR, HTT MAPT 1/4885ALOX15 1017/4885MEN1 2502/4885
US-20110312926-A1 2-(N-Substituted Piperazinyl) Steroid Derivatives NR5A1, HSD17B11, CYP17A1 MAPT 4699/4885ALOX15 2932/4885MEN1 3323/4885
US-11174282-B2 Aminosteroid derivatives and process for producing same HSD17B11, HSD17B7, CYP19A1 MAPT 3922/4885ALOX15 1313/4885MEN1 1439/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.