SCHEMBL8485083

SCHEMBL8485083

CNC(=O)C(CNC(=O)OC(C)(C)C)c1ccc(-c2cccc3ccccc23)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PPARG P37231 9/20 0.43
PPARA Q07869 9/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
PPARD Q03181 1/20 0.43
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
MMP2 P08253 1/20 0.41
MMP3 P08254 1/20 0.41
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NQO2 P16083 1/20 0.39
MALT1 Q9UDY8 1/20 0.38
KDM4A O75164 1/20 0.37
SYK P43405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6575223 0.80 CTSS (0.46) CTSSCTSKNQO2KDM4ASYK
SCHEMBL22002108 0.79 SYK (0.40) PPARGPPARACTSSCTSKSYK
SCHEMBL20860285 0.77 FFAR2 (0.44) PPARGPPARACTSSCTSKSYK
SCHEMBL8485076 0.77 CTSS (0.57) PPARGPPARACYP2C9CYP2C19PPARD
SCHEMBL22703144 0.74 PPARG (0.44) PPARGPPARACYP2C9CYP2C19PPARD
SCHEMBL22703156 0.74 PPARG (0.44) PPARGPPARACYP2C9CYP2C19PPARD
SCHEMBL27414019 0.74 CTSS (0.48) PPARGPPARACTSSCTSKMALT1
SCHEMBL6827827 0.73 PTPRB (0.45)
SCHEMBL6831591 0.73 NPC1 (0.45) PPARGPPARAMMP2
SCHEMBL6831647 0.73 PTPRB (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5986132-A Synthesis of carboxylic acid derivatives BRITISH BIOTECH PHARMACEUTICALS LTD. (GB) 1999-11-16 US disclosed