SCHEMBL8485285

SCHEMBL8485285

CCCCCC(=O)Oc1c(C)c(OC)cc2c1COC(C)C2

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
F3 P13726 1/20 0.42
TOP2A P11388 1/20 0.36
NLRP3 Q96P20 1/20 0.36
CYP3A4 P08684 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
EPHX2 P34913 1/20 0.35
TRPV1 Q8NER1 5/20 0.35
ALOX15 P16050 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8485766 0.99 F3 (0.41) F3TOP2ANLRP3CYP3A4MAPK1
SCHEMBL8485869 0.99 F3 (0.41) F3TOP2ANLRP3CYP3A4MAPK1
SCHEMBL8482088 0.97 F3 (0.39) F3TOP2ANLRP3CYP3A4MAPK1
SCHEMBL8485301 0.93 ALDH1A1 (0.35) F3NLRP3KDM4EALDH1A1GAA
SCHEMBL8487162 0.92 F3 (0.38) F3TOP2ANLRP3CYP3A4MAPK1
SCHEMBL8479256 0.91 TOP2A (0.38) F3TOP2ANLRP3CYP3A4MAPK1
SCHEMBL8483878 0.91 TOP2A (0.38) F3TOP2ANLRP3CYP3A4MAPK1
SCHEMBL8483098 0.91 TOP2A (0.38) F3TOP2ANLRP3CYP3A4MAPK1
SCHEMBL8483236 0.84 LMNA (0.36) NLRP3CYP3A4MAPK1CYP2C19ALOX15
SCHEMBL8486293 0.82 POLB (0.39) F3CYP3A4KDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922889-A REACTING 3,7-DIMETHYL-6,8-DIMETHOXYISOCHROMAN WITH SODIUM ETHYL THIOLATE OR SODIUM HYDRIDE TO PRODUCE 3,7-DIMETHYL-6-HYDROXY-8-METHOXYISOCHROMAN; POSSESS PHYTOTOXIC ACTIVITY USED AS A BIODEGRADABLE HERBICIDE THE UNITED STATES OD AMERICA AS REPRESENTED BY THE SECRETARY OF AGRICULTURE (US) 1999-07-13 US claimed
US-5922889-A REACTING 3,7-DIMETHYL-6,8-DIMETHOXYISOCHROMAN WITH SODIUM ETHYL THIOLATE OR SODIUM HYDRIDE TO PRODUCE 3,7-DIMETHYL-6-HYDROXY-8-METHOXYISOCHROMAN; POSSESS PHYTOTOXIC ACTIVITY USED AS A BIODEGRADABLE HERBICIDE THE UNITED STATES OD AMERICA AS REPRESENTED BY THE SECRETARY OF AGRICULTURE (US) 1999-07-13 US disclosed