SCHEMBL8485494

SCHEMBL8485494

COCc1ccccc1CCNc1ncnc2c(C)cccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 5/20 0.47
AURKA O14965 4/20 0.47
LDHA P00338 1/20 0.45
PDPK1 O15530 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPK1 P28482 5/20 0.42
TSHR P16473 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
ALOX15 P16050 1/20 0.42
CYP2C19 P33261 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
HTT P42858 5/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HPGD P15428 1/20 0.41
APP P05067 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9609099 0.88 RPS6KB1 (0.52) RPS6KB1AURKALDHAPDPK1ALDH1A1
SCHEMBL8491743 0.87 RPS6KB1 (0.46) RPS6KB1AURKALDHAPDPK1ALDH1A1
SCHEMBL8504575 0.87 RPS6KB1 (0.46) RPS6KB1AURKALDHAPDPK1ALDH1A1
SCHEMBL8484113 0.86 HTT (0.42) LDHAALDH1A1KDM4EMAPK1TSHR
SCHEMBL8490466 0.85 RPS6KB1 (0.49) RPS6KB1AURKALDHAPDPK1ALDH1A1
SCHEMBL8483456 0.84 RXFP1 (0.42) LDHAALDH1A1KDM4EMAPK1TSHR
SCHEMBL9608188 0.82 AURKA (0.42) RPS6KB1AURKALDHAALDH1A1KDM4E
SCHEMBL5569127 0.81 MEN1 (0.48) RPS6KB1AURKAALDH1A1KDM4EMAPK1
SCHEMBL8484236 0.80 LDHA (0.46) LDHAALDH1A1KDM4EMAPK1TSHR
SCHEMBL8482247 0.79 MAPT (0.42) LDHAALDH1A1KDM4EMAPK1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2455371-A1 4-(3-BUTYNYL)AMINOPYRIMIDINE DERIVATIVES AS PEST CONTROL AGENTS FOR AGRICULTURAL AND HORTICULTURAL USE SDS Biotech K. K. (JP) 2012-05-23 EP disclosed