SCHEMBL8485649

SCHEMBL8485649

CCCCCCCCN(CC(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1)S(C)(=O)=O

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PER2 O15055 7/20 0.40
S1PR1 P21453 1/20 0.39
CRY1 Q16526 6/20 0.38
CRY2 Q49AN0 6/20 0.38
KDM4E B2RXH2 1/20 0.36
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
ALOX15 P16050 1/20 0.36
BACE1 P56817 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8490612 1.00 PER2 (0.40) PER2S1PR1CRY1CRY2KDM4E
SCHEMBL8489932 0.95 PER2 (0.42) PER2S1PR1CRY1CRY2KDM4E
SCHEMBL8488600 0.86 PER2 (0.38) PER2CRY1CRY2KDM4EUSP2
SCHEMBL8487214 0.86 PER2 (0.38) PER2CRY1CRY2KDM4EUSP2
SCHEMBL9004290 0.86 PER2 (0.38) PER2CRY1CRY2BACE1
SCHEMBL8486390 0.85 S1PR1 (0.36) PER2S1PR1CRY1CRY2
SCHEMBL8489654 0.85 S1PR1 (0.36) PER2S1PR1CRY1CRY2
SCHEMBL8488753 0.83 PER2 (0.51) PER2CRY1CRY2KDM4EALDH1A1
SCHEMBL9004350 0.82 MAPT (0.37) PER2CRY1CRY2BACE1
SCHEMBL8491767 0.81 PER2 (0.39) PER2CRY1CRY2KDM4EUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919431-A 1,4,7,10-tetraazacyclododecane derivatives, their use, pharmaceutical agents containing these compounds and process for their production SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-06 US disclosed