SCHEMBL8488753

SCHEMBL8488753

COCCN(CC(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(=O)O)CC1)S(C)(=O)=O

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PER2 O15055 10/20 0.51
CRY1 Q16526 9/20 0.51
CRY2 Q49AN0 9/20 0.51
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 1/20 0.36
BACE1 P56817 4/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8491775 0.86 PER2 (0.47) PER2CRY1CRY2ALDH1A1KDM4E
SCHEMBL9004290 0.86 PER2 (0.38) PER2CRY1CRY2BACE1L3MBTL1
SCHEMBL8488046 0.85 PER2 (0.42) PER2CRY1CRY2
SCHEMBL8489932 0.85 PER2 (0.42) PER2CRY1CRY2ALDH1A1KDM4E
SCHEMBL8490612 0.83 PER2 (0.40) PER2CRY1CRY2ALDH1A1KDM4E
SCHEMBL8485649 0.83 PER2 (0.40) PER2CRY1CRY2ALDH1A1KDM4E
SCHEMBL9004350 0.82 MAPT (0.37) PER2CRY1CRY2BACE1L3MBTL1
SCHEMBL9004320 0.82 PER2 (0.46) PER2CRY1CRY2ALDH1A1BACE1
SCHEMBL8488572 0.80 BACE1 (0.48) PER2CRY1CRY2ALDH1A1KDM4E
SCHEMBL21618562 0.77 ALDH1A1 (0.44) ALDH1A1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5919431-A 1,4,7,10-tetraazacyclododecane derivatives, their use, pharmaceutical agents containing these compounds and process for their production SCHERING AKTIENGESELLSCHAFT (DE) 1999-07-06 US disclosed